| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1766081 | 1 | PPB | 99.21 | % | ALA3301365 | % | |||||
| 2. | ALA1766081 | 1 | PPB | 98.51 | % | ALA3301368 | % | |||||
| 3. | ALA1766081 | 1 | LogD7.4 | 3.8 | ALA3301363 | |||||||
| 4. | ALA1766081 | 1 | PPB | 96.87 | % | ALA3301366 | % | |||||
| 5. | ALA1766081 | 1 | solubility | = | 15.9 | mg/ml | ALA1953654 | ug.mL-1 | ||||
| 6. | ALA1766081 | 1 | solubility | = | 15.9 | mg/ml | ALA1953653 | ug.mL-1 | ||||
| 7. | ALA1766081 | 1 | Intrinsic activity | = | 89 | % | ALA1953652 | % | Rattus norvegicus | |||
| 8. | ALA1766081 | 1 | Intrinsic activity | = | 37 | % | ALA1953651 | % | Homo sapiens | |||
| 9. | ALA1766081 | 1 | EC50 | = | 83 | nM | ALA1953650 | 7.08 | nM | Rattus norvegicus | ||
| 10. | ALA1766081 | 1 | EC50 | = | 7.3 | nM | ALA1953649 | 8.14 | nM | Homo sapiens | ||
| 11. | ALA1766081 | 1 | EC50 | = | 15 | nM | ALA1781103 | 7.82 | nM | Homo sapiens | ||
| 12. | ALA1766081 | 1 | Ki | = | 140 | nM | ALA1769550 | 6.85 | nM | Rattus norvegicus | ||
| 13. | ALA1766081 | 1 | solubility | > | 40 | mg/ml | ALA1769450 | ug.mL-1 | ||||
| 14. | ALA1766081 | 1 | CL | = | 15 | ml/min.kg | ALA1769447 | mL.min-1.kg-1 | Homo sapiens | |||
| 15. | ALA1766081 | 1 | Ki | = | 23 | nM | ALA1769549 | 7.64 | nM | Homo sapiens | ||
| 16. | ALA1766081 | 1 | Intrinsic activity | = | 21 | % | ALA1769546 | % | Homo sapiens | |||
| 17. | ALA1766081 | 1 | EC50 | = | 14 | nM | ALA1769445 | 7.85 | nM | Homo sapiens | ||
| 18. | ALA1766081 | 1 | Intrinsic activity | = | 70 | % | ALA1769547 | % | Rattus norvegicus | |||
| 19. | ALA1766081 | 1 | EC50 | = | 84 | nM | ALA1769446 | 7.08 | nM | Rattus norvegicus |
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