| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1770317 | 6b | Papp | 0 | ALA4689783 | Not Determined | ||||||
| 2. | ALA1770317 | 6b | Kinetic_solubility | 0 | ALA4689782 | Not Determined | ||||||
| 3. | ALA1770317 | 6b | Kinetic_solubility | 0 | ALA4689781 | Not Determined | ||||||
| 4. | ALA1770317 | 6b | t1/2 | 0 | ALA4689780 | Not Determined | ||||||
| 5. | ALA1770317 | 6b | t1/2 | 0 | ALA4689779 | Not Determined | ||||||
| 6. | ALA1770317 | 6b | IC50 | = | 68 | nM | ALA4689778 | 7.17 | nM | Homo sapiens | ||
| 7. | ALA1770317 | 6b | Ki | = | 10 | nM | ALA4689777 | 8.00 | nM | Homo sapiens | ||
| 8. | ALA1770317 | 6b | Activity | 0 | ALA1771838 | Active | ||||||
| 9. | ALA1770317 | 6b | Activity | 0 | ALA1771839 | Active | Rattus norvegicus | |||||
| 10. | ALA1770317 | 6b | F | = | 100 | % | ALA1771837 | % | Rattus norvegicus | |||
| 11. | ALA1770317 | 6b | AUC | = | 4.4 | microg.hr/mL | ALA1771836 | ng.hr.mL-1 | Rattus norvegicus | |||
| 12. | ALA1770317 | 6b | t1/2 | = | 3.5 | hr | ALA1771835 | hr | Rattus norvegicus | |||
| 13. | ALA1770317 | 6b | CL | = | 5.1 | ml/min.kg | ALA1771834 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 14. | ALA1770317 | 6b | pKi | = | 8 | ALA1771833 | 8.00 | nM | Homo sapiens | |||
| 15. | ALA1770317 | 6b | pKi | = | 8 | ALA2039059 | 8.00 | nM | Homo sapiens | |||
| 16. | ALA1770317 | 6b | pKi | = | 8 | ALA2039058 | 8.00 | nM | Rattus norvegicus | |||
| 17. | ALA1770317 | 6b | pKi | < | 4.3 | ALA2039030 | nM | Homo sapiens | ||||
| 18. | ALA1770317 | 6b | pKi | = | 7.7 | ALA2039031 | 7.70 | nM | ||||
| 19. | ALA1770317 | 6b | pKi | = | 8.3 | ALA2039039 | 8.30 | nM | Homo sapiens | |||
| 20. | ALA1770317 | 6b | t1/2 | = | 4 | hr | ALA2039040 | hr | Rattus norvegicus |
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