# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1774023 | 47 | Ratio | > | 2 | ALA1810828 | Homo sapiens | |||||
2. | ALA1774023 | 47 | Papp | < | 100 | nm/s | ALA1810827 | nm/s | Homo sapiens | |||
3. | ALA1774023 | 47 | CL | = | 42 | microL/min/mg | ALA1810826 | mL.min-1.g-1 | Rattus norvegicus | |||
4. | ALA1774023 | 47 | CL | < | 12 | microL/min/mg | ALA1810825 | mL.min-1.g-1 | Homo sapiens | |||
5. | ALA1774023 | 47 | pKi | = | 7.66 | ALA1810823 | 7.66 | nM | Rattus norvegicus | |||
6. | ALA1774023 | 47 | pKi | = | 9.63 | ALA1810552 | 9.63 | nM | Homo sapiens | |||
7. | ALA1774023 | 47 | Activity | = | 58 | % | ALA1776947 | % | Rattus norvegicus | |||
8. | ALA1774023 | 47 | Activity | = | 77.4 | % | ALA1776946 | % | Rattus norvegicus | |||
9. | ALA1774023 | 47 | pKi | <= | 5 | ALA1776945 | nM | Homo sapiens | ||||
10. | ALA1774023 | 47 | pKi | <= | 5 | ALA1776944 | nM | Homo sapiens | ||||
11. | ALA1774023 | 47 | pKi | <= | 5 | ALA1776943 | nM | Homo sapiens | ||||
12. | ALA1774023 | 47 | pKi | = | 5.38 | ALA1776942 | 5.38 | nM | Homo sapiens | |||
13. | ALA1774023 | 47 | pIC50 | = | 7.26 | ALA1776941 | 7.26 | nM | Homo sapiens | |||
14. | ALA1774023 | 47 | CL | = | 16 | ml/min.kg | ALA1776940 | mL.min-1.kg-1 | Rattus norvegicus | |||
15. | ALA1774023 | 47 | CL | < | 12 | microL/min/mg | ALA1776763 | mL.min-1.g-1 | Homo sapiens | |||
16. | ALA1774023 | 47 | CL | = | 42 | microL/min/mg | ALA1776930 | mL.min-1.g-1 | Rattus norvegicus | |||
17. | ALA1774023 | 47 | pKi | = | 9.63 | ALA1776931 | 9.63 | nM | Homo sapiens | |||
18. | ALA1774023 | 47 | pKi | = | 7.66 | ALA1776932 | 7.66 | nM | Rattus norvegicus | |||
19. | ALA1774023 | 47 | F | < | 1 | % | ALA1776935 | % | Rattus norvegicus | |||
20. | ALA1774023 | 47 | t1/2 | = | 11.5 | hr | ALA1776936 | hr | Rattus norvegicus |