# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1774024 | 48 | Activity | = | 50 | % | ALA1776948 | % | Rattus norvegicus | |||
2. | ALA1774024 | 48 | pKi | <= | 5 | ALA1776945 | nM | Homo sapiens | ||||
3. | ALA1774024 | 48 | pKi | <= | 5 | ALA1776944 | nM | Homo sapiens | ||||
4. | ALA1774024 | 48 | pKi | <= | 5 | ALA1776943 | nM | Homo sapiens | ||||
5. | ALA1774024 | 48 | pKi | = | 5.8 | ALA1776942 | 5.80 | nM | Homo sapiens | |||
6. | ALA1774024 | 48 | pIC50 | = | 7.43 | ALA1776941 | 7.43 | nM | Homo sapiens | |||
7. | ALA1774024 | 48 | CL | = | 44 | ml/min.kg | ALA1776940 | mL.min-1.kg-1 | Rattus norvegicus | |||
8. | ALA1774024 | 48 | CL | = | 58 | microL/min/mg | ALA1776763 | mL.min-1.g-1 | Homo sapiens | |||
9. | ALA1774024 | 48 | CL | = | 55 | microL/min/mg | ALA1776930 | mL.min-1.g-1 | Rattus norvegicus | |||
10. | ALA1774024 | 48 | pKi | = | 9.25 | ALA1776931 | 9.25 | nM | Homo sapiens | |||
11. | ALA1774024 | 48 | pKi | = | 8.38 | ALA1776932 | 8.38 | nM | Rattus norvegicus | |||
12. | ALA1774024 | 48 | F | = | 4 | % | ALA1776935 | % | Rattus norvegicus | |||
13. | ALA1774024 | 48 | t1/2 | = | 8.2 | hr | ALA1776936 | hr | Rattus norvegicus | |||
14. | ALA1774024 | 48 | Cmax | = | 19 | ng/ml | ALA1776937 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
15. | ALA1774024 | 48 | Tmax | = | 3.5 | hr | ALA1776938 | hr | Rattus norvegicus | |||
16. | ALA1774024 | 48 | Vdss | = | 17.7 | L/Kg | ALA1776939 | L.kg-1 | Rattus norvegicus |