# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1779978 | 6, PF-04399482-00 | t1/2 | = | 5.76 | min | ALA1780344 | hr | Homo sapiens | |||
2. | ALA1779978 | 6, PF-04399482-00 | CL | = | 158 | microL/min/mg | ALA1780338 | mL.min-1.g-1 | Homo sapiens | |||
3. | ALA1779978 | 6, PF-04399482-00 | Selectivity ratio | > | 1000 | ALA1780337 | ||||||
4. | ALA1779978 | 6, PF-04399482-00 | Selectivity ratio | > | 1000 | ALA1780336 | ||||||
5. | ALA1779978 | 6, PF-04399482-00 | Selectivity ratio | > | 1000 | ALA1780335 | ||||||
6. | ALA1779978 | 6, PF-04399482-00 | Selectivity ratio | > | 1000 | ALA1780334 | ||||||
7. | ALA1779978 | 6, PF-04399482-00 | IC50 | = | 240 | nM | ALA1780332 | 6.62 | nM | Homo sapiens | ||
8. | ALA1779978 | 6, PF-04399482-00 | IC50 | = | 1.8 | nM | ALA1780333 | 8.74 | nM | Homo sapiens |