# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1783734 | 2 | Stability | = | 85 | % | ALA3768926 | % | ||||
2. | ALA1783734 | 2 | Activity | = | 4.39 | mM | ALA3768924 | mM | Mus musculus | |||
3. | ALA1783734 | 2 | Activity | = | 2.83 | mM | ALA3768923 | mM | Mus musculus | |||
4. | ALA1783734 | 2 | EC50 | = | 6.32 | uM | ALA3768919 | 5.20 | nM | Homo sapiens | ||
5. | ALA1783734 | 2 | Emax | = | 716.4 | % | ALA3768920 | % | Homo sapiens | |||
6. | ALA1783734 | 2 | LogD7.4 | 1.39 | ALA3301363 | |||||||
7. | ALA1783734 | 2 | Solubility | 1148.2 | uM | ALA3301364 | nM | |||||
8. | ALA1783734 | 2 | TI | < | 5 | ALA3583645 | ||||||
9. | ALA1783734 | 2 | Activity | < | 60 | mg/dl | ALA3583644 | mg/dl | Rattus norvegicus | |||
10. | ALA1783734 | 2 | Activity | > | 20 | % | ALA3583542 | % | Rattus norvegicus | |||
11. | ALA1783734 | 2 | EC50 | = | 364 | nM | ALA3583541 | 6.44 | nM | Homo sapiens | ||
12. | ALA1783734 | 2 | Kd | = | 218.4 | nM | ALA3583540 | 6.66 | nM | Homo sapiens | ||
13. | ALA1783734 | 2 | K | = | 43.9 | 10'-3/s | ALA3583539 | 10'-3/s | Homo sapiens | |||
14. | ALA1783734 | 2 | K | = | 2.05 | 10'5/M/s | ALA3583538 | 10'5/M/s | Homo sapiens | |||
15. | ALA1783734 | 2 | t1/2 | = | 15.8 | s | ALA3582523 | hr | Homo sapiens | |||
16. | ALA1783734 | 2 | Activity | 0 | ALA4272669 | Active | Mus musculus | |||||
17. | ALA1783734 | 2 | Ratio AUC | = | 2.9 | ALA4272700 | ||||||
18. | ALA1783734 | 2 | Ratio AUC | = | 3.1 | ALA4272698 | ||||||
19. | ALA1783734 | 2 | Ratio AUC | = | 3.2 | ALA4272697 | ||||||
20. | ALA1783734 | 2 | Ratio AUC | = | 1.4 | ALA4272696 |