| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1784577 | 32, DSM190 | Ratio IC50 | = | 100 | ALA3297103 | ||||||
| 2. | ALA1784577 | 32, DSM190 | IC50 | > | 30 | uM | ALA3296344 | nM | Mus musculus | |||
| 3. | ALA1784577 | 32, DSM190 | IC50 | > | 100 | uM | ALA3296349 | nM | ||||
| 4. | ALA1784577 | 32, DSM190 | IC50 | > | 100 | uM | ALA3296347 | nM | Homo sapiens | |||
| 5. | ALA1784577 | 32, DSM190 | IC50 | = | 37 | uM | ALA3296348 | 4.43 | nM | Rattus norvegicus | ||
| 6. | ALA1784577 | 32, DSM190 | IC50 | = | 190 | nM | ALA3705388 | 6.72 | 318875 | nM | Plasmodium falciparum (isolate 3D7) | |
| 7. | ALA1784577 | 32, DSM190 | solubility | = | 9 | uM | ALA1785549 | nM | ||||
| 8. | ALA1784577 | 32, DSM190 | logD | = | 2.9 | ALA1785548 | ||||||
| 9. | ALA1784577 | 32, DSM190 | PPB | = | 97.3 | % | ALA1785553 | % | Rattus norvegicus | |||
| 10. | ALA1784577 | 32, DSM190 | Activity | 0 | ALA1785739 | Non-toxic | Rattus norvegicus | |||||
| 11. | ALA1784577 | 32, DSM190 | Activity | 0 | ALA1785738 | Non-toxic | Rattus norvegicus | |||||
| 12. | ALA1784577 | 32, DSM190 | Activity | 0 | ALA1785556 | Non-toxic | Mus musculus | |||||
| 13. | ALA1784577 | 32, DSM190 | Ratio | = | 10 | ALA1785546 | ||||||
| 14. | ALA1784577 | 32, DSM190 | EC50 | = | 0.22 | uM | ALA1785545 | 6.66 | nM | Plasmodium falciparum | ||
| 15. | ALA1784577 | 32, DSM190 | IC50 | = | 0.19 | uM | ALA1785541 | 6.72 | nM | Plasmodium falciparum | ||
| 16. | ALA1784577 | 32, DSM190 | IC50 | = | 0.28 | uM | ALA1785542 | 6.55 | nM | |||
| 17. | ALA1784577 | 32, DSM190 | IC50 | > | 30 | uM | ALA1785543 | nM | Homo sapiens | |||
| 18. | ALA1784577 | 32, DSM190 | EC50 | = | 1.1 | uM | ALA1785544 | 5.96 | nM | Plasmodium falciparum | ||
| 19. | ALA1784577 | 32, DSM190 | F | > | 100 | % | ALA1785737 | % | Rattus norvegicus | |||
| 20. | ALA1784577 | 32, DSM190 | AUC | = | 75007 | uM.min | ALA1785735 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus |
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