# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA12858 | 3 | Ratio | = | 0.7 | ALA849573 | Homo sapiens | |||||
2. | ALA12858 | 3 | Ratio | = | 8.3 | ALA848595 | Homo sapiens | |||||
3. | ALA12858 | 3 | Lethal dose | = | 60 | mg kg-1 | ALA722392 | mg kg-1 | Mus musculus | |||
4. | ALA12858 | 3 | Change | = | 86 | % | ALA735378 | % | Mus musculus | |||
5. | ALA12858 | 3 | Ileal activity | < | 0.01 | uM | ALA787630 | uM | Rattus norvegicus | |||
6. | ALA12858 | 3 | IC50 | = | 0.47 | uM | ALA744480 | 6.33 | nM | Mus musculus | ||
7. | ALA12858 | 3 | IC50 | = | 0.66 | uM | ALA745515 | 6.18 | nM | Mus musculus | ||
8. | ALA12858 | 3 | IC50 | = | 2.4 | uM | ALA659267 | 5.62 | nM | Homo sapiens | ||
9. | ALA12858 | 3 | IC50 | = | 0.29 | uM | ALA641506 | 6.54 | nM | Homo sapiens |