# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1802187 | 16b | log Pe | = | -4.6 | ALA1805241 | ||||||
2. | ALA1802187 | 16b | AUC | = | 21.69 | ug.hr/ml | ALA1805480 | ng.hr.mL-1 | ||||
3. | ALA1802187 | 16b | AUC | = | 2.1 | ug.hr/ml | ALA1805064 | ng.hr.mL-1 | Mus musculus | |||
4. | ALA1802187 | 16b | AUC | = | 1.89 | ug.hr/ml | ALA1805327 | ng.hr.mL-1 | ||||
5. | ALA1802187 | 16b | AUC | = | 1.02 | ug.hr/ml | ALA1805326 | ng.hr.mL-1 | Mus musculus | |||
6. | ALA1802187 | 16b | Stability | 0 | ALA1805247 | Unstable | % | Mus musculus | ||||
7. | ALA1802187 | 16b | Stability | 0 | ALA1805248 | Stable | % | Mus musculus | ||||
8. | ALA1802187 | 16b | Therm_solubility | = | 11.9 | ug ml-1 | ALA1805244 | ug.mL-1 | ||||
9. | ALA1802187 | 16b | Stability | = | 80 | % | ALA1805246 | % | ||||
10. | ALA1802187 | 16b | Stability | = | 80 | % | ALA1805245 | % | ||||
11. | ALA1802187 | 16b | Ratio IC50 | = | 0.06 | ALA1805066 | Escherichia coli K-12 | |||||
12. | ALA1802187 | 16b | PPB | = | 94 | % | ALA1805250 | % | Homo sapiens | |||
13. | ALA1802187 | 16b | permeability | = | 41 | % | ALA1805242 | % | ||||
14. | ALA1802187 | 16b | Papp | = | 2.05 | 10'-6 cm/s | ALA1805243 | 10'-6 cm/s | Homo sapiens | |||
15. | ALA1802187 | 16b | logD | = | 2.32 | ALA1805240 | ||||||
16. | ALA1802187 | 16b | IC50 | = | 4.8 | nM | ALA1805065 | 8.32 | nM | Escherichia coli K-12 | ||
17. | ALA1802187 | 16b | IC50 | = | 9 | uM | ALA1805067 | 5.05 | nM | Escherichia coli K-12 |