# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | LM10 | 58 | IC50 | > | 400 | uM | ALA3630809 | nM | Mus musculus | |||
2. | LM10 | 58 | IC50 | = | 1.96 | uM | ALA3630808 | 5.71 | nM | Mus musculus | ||
3. | LM10 | 58 | IC50 | = | 0.62 | uM | ALA3630807 | 6.21 | nM | Homo sapiens | ||
4. | LM10 | 58 | Ki | = | 5.6 | uM | ALA4383521 | 5.25 | nM | Homo sapiens | ||
5. | LM10 | 58 | IC50 | = | 0.398 | uM | ALA4383519 | 6.40 | nM | Homo sapiens | ||
6. | LM10 | 58 | IC50 | = | 0.671 | uM | ALA4383518 | 6.17 | nM | Homo sapiens | ||
7. | LM10 | 58 | Ki | = | 7.47 | uM | ALA4383516 | 5.13 | nM | Homo sapiens | ||
8. | LM10 | 58 | IC50 | = | 18.7 | uM | ALA4383515 | 4.73 | nM | Homo sapiens | ||
9. | LM10 | 58 | Ki | = | 5.5 | uM | ALA4370865 | 5.26 | nM | Homo sapiens | ||
10. | LM10 | 58 | Drug metabolism | 0 | ALA4810622 | Metabolite_Detected | ||||||
11. | LM10 | 58 | Drug metabolism | 0 | ALA4810621 | Metabolite_Detected | ||||||
12. | LM10 | 58 | INH | 0 | ALA4810620 | Not Active | % | Homo sapiens | ||||
13. | LM10 | 58 | INH | 0 | ALA4810619 | Not Active | % | Homo sapiens | ||||
14. | LM10 | 58 | t1/2 | > | 1440 | min | ALA4810618 | hr | ||||
15. | LM10 | 58 | LD50 | > | 100 | uM | ALA4810617 | uM | Mus musculus | |||
16. | LM10 | 58 | IC50 | = | 1.74 | uM | ALA4810616 | 5.76 | nM | Homo sapiens | ||
17. | LM10 | 58 | IC50 | = | 6.1 | uM | ALA4810615 | 5.21 | nM | Homo sapiens | ||
18. | LM10 | 58 | IC50 | = | 11.58 | uM | ALA4620359 | 4.94 | nM | Homo sapiens | ||
19. | LM10 | 58 | IC50 | 0 | ALA4620353 | Not Determined | Homo sapiens | |||||
20. | LM10 | 58 | CC50 | > | 20 | uM | ALA4296191 | Median N= 2; Maxinhib 15.4 Pct | nM | Homo sapiens |