| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1828889 | 5 | BPR | = | 6.2 | ALA1833638 | ||||||
| 2. | ALA1828889 | 5 | F | = | 16 | % | ALA1833637 | % | Rattus norvegicus | |||
| 3. | ALA1828889 | 5 | Vdss | = | 14423 | ml/kg | ALA1833636 | L.kg-1 | Rattus norvegicus | |||
| 4. | ALA1828889 | 5 | t1/2 | = | 3.4 | hr | ALA1833635 | hr | Rattus norvegicus | |||
| 5. | ALA1828889 | 5 | t1/2 | = | 1.7 | hr | ALA1833634 | hr | Rattus norvegicus | |||
| 6. | ALA1828889 | 5 | CL | = | 186 | ml/min.kg | ALA1833633 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 7. | ALA1828889 | 5 | Cmax | = | 27.4 | ng/ml | ALA1833632 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 8. | ALA1828889 | 5 | Tmax | = | 4 | hr | ALA1833631 | hr | Rattus norvegicus | |||
| 9. | ALA1828889 | 5 | AUC | = | 153 | ng.hr/ml | ALA1833630 | ng.hr.mL-1 | Rattus norvegicus | |||
| 10. | ALA1828889 | 5 | AUC | = | 96 | ng.hr/ml | ALA1833629 | ng.hr.mL-1 | Rattus norvegicus | |||
| 11. | ALA1828889 | 5 | Activity | 0 | ALA1833628 | Active | Rattus norvegicus | |||||
| 12. | ALA1828889 | 5 | EC50 | = | 81 | nM | ALA1833627 | 7.09 | nM | Rattus norvegicus | ||
| 13. | ALA1828889 | 5 | EC50 | = | 4 | nM | ALA1833626 | 8.40 | nM | Homo sapiens | ||
| 14. | ALA1828889 | 5 | IC50 | = | 8 | nM | ALA1833625 | 8.10 | nM | Homo sapiens |
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