# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1829763 | 25f | IC50 | = | 0.8 | nM | ALA5245459 | 9.10 | nM | Homo sapiens | ||
2. | ALA1829763 | 25f | CLint | < | 3 | microL/min/1E6 cells | ALA3301371 | uL.min-1.(10^6cells)-1 | ||||
3. | ALA1829763 | 25f | Solubility | 2.5 | uM | ALA3301364 | nM | |||||
4. | ALA1829763 | 25f | CLint | 14.13 | microL/min/mg | ALA3301370 | mL.min-1.g-1 | |||||
5. | ALA1829763 | 25f | solubility | 0 | ALA4036193 | Bld | ||||||
6. | ALA1829763 | 25f | Ratio IC50 | > | 1000 | ALA4036214 | ||||||
7. | ALA1829763 | 25f | Ratio IC50 | > | 1000 | ALA4036213 | ||||||
8. | ALA1829763 | 25f | Ratio IC50 | > | 1000 | ALA4036212 | ||||||
9. | ALA1829763 | 25f | PPB | > | 99 | % | ALA4036210 | % | Homo sapiens | |||
10. | ALA1829763 | 25f | logP | = | 4.2 | ALA4036209 | ||||||
11. | ALA1829763 | 25f | IC80 | > | 1 | uM | ALA4036199 | uM | Homo sapiens | |||
12. | ALA1829763 | 25f | IC50 | = | 2.5 | nM | ALA4036190 | 8.60 | nM | Homo sapiens | ||
13. | ALA1829763 | 25f | IC50 | = | 0.8 | nM | ALA4036189 | 9.10 | nM | Homo sapiens | ||
14. | ALA1829763 | 25f | IC50 | = | 17.74 | nM | ALA3705551 | 7.75 | 228062 | nM | Homo sapiens | |
15. | ALA1829763 | 25f | IC50 | = | 0.75 | nM | ALA3705551 | 9.12 | 228042 | nM | Homo sapiens | |
16. | ALA1829763 | 25f | IC50 | = | 17.74 | nM | ALA3705119 | 7.75 | 227384 | nM | Homo sapiens | |
17. | ALA1829763 | 25f | IC50 | = | 0.75 | nM | ALA3705121 | 9.12 | 227297 | nM | Homo sapiens | |
18. | ALA1829763 | 25f | IC50 | = | 4900 | nM | ALA3705153 | 5.31 | 226958 | nM | Homo sapiens | |
19. | ALA1829763 | 25f | IC50 | = | 5700 | nM | ALA3705156 | 5.24 | 226944 | nM | Homo sapiens | |
20. | ALA1829763 | 25f | IC50 | = | 4100 | nM | ALA3705155 | 5.39 | 226925 | nM | Homo sapiens |