# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA166 | melarsoprol | IC50 | = | 0.011 | uM | ALA2445916 | 7.96 | nM | Trypanosoma brucei rhodesiense | ||
2. | ALA166 | melarsoprol | IC50 | = | 0.005 | uM | ALA2438768 | 8.30 | nM | Trypanosoma brucei rhodesiense | ||
3. | ALA166 | melarsoprol | Activity | 0 | ALA2422947 | Active | Trypanosoma brucei rhodesiense | |||||
4. | ALA166 | melarsoprol | IC50 | = | 0.006 | uM | ALA2422962 | 8.22 | nM | Trypanosoma brucei rhodesiense | ||
5. | ALA166 | melarsoprol | IC50 | = | 7.78 | mM | ALA2422955 | nM | Rattus norvegicus | |||
6. | ALA166 | melarsoprol | MSD | > | 60 | day | ALA2422953 | day | Trypanosoma brucei rhodesiense | |||
7. | ALA166 | melarsoprol | Ratio IC50 | = | 1222 | ALA2422961 | ||||||
8. | ALA166 | melarsoprol | IC50 | = | 4 | nM | ALA2421064 | 8.40 | nM | Trypanosoma brucei rhodesiense | ||
9. | ALA166 | melarsoprol | IC50 | = | 0.009 | uM | ALA2416704 | 8.05 | nM | Trypanosoma brucei rhodesiense | ||
10. | ALA166 | melarsoprol | IC50 | = | 7.78 | uM | ALA2416702 | 5.11 | nM | Rattus norvegicus | ||
11. | ALA166 | melarsoprol | Ratio IC50 | = | 1945 | ALA2416701 | ||||||
12. | ALA166 | melarsoprol | IC50 | = | 0.005 | uM | ALA2411135 | 8.30 | nM | Trypanosoma brucei rhodesiense | ||
13. | ALA166 | melarsoprol | Ratio IC50 | = | 10 | ALA2404683 | Trypanosoma brucei brucei | |||||
14. | ALA166 | melarsoprol | MSD | > | 60 | day | ALA2399211 | day | Trypanosoma brucei rhodesiense | |||
15. | ALA166 | melarsoprol | IC50 | = | 0.004 | uM | ALA2399341 | 8.40 | nM | Trypanosoma brucei rhodesiense | ||
16. | ALA166 | melarsoprol | IC50 | = | 5.12 | uM | ALA2399214 | 5.29 | nM | Rattus norvegicus | ||
17. | ALA166 | melarsoprol | Ratio IC50 | = | 1275 | ALA2399340 | ||||||
18. | ALA166 | melarsoprol | Activity | 0 | ALA2399215 | Active | Trypanosoma brucei rhodesiense | |||||
19. | ALA166 | melarsoprol | IC50 | = | 0.008 | uM | ALA2390652 | 8.12 | nM | Trypanosoma brucei rhodesiense | ||
20. | ALA166 | melarsoprol | Ratio IC50 | = | 1 | ALA2072690 | Trypanosoma brucei brucei |