# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA166 | melarsoprol | IC50 | = | 0.007 | uM | ALA4416651 | 8.15 | nM | Trypanosoma brucei rhodesiense | ||
2. | ALA166 | melarsoprol | Ratio IC50 | = | 3284.1 | ALA4413423 | ||||||
3. | ALA166 | melarsoprol | CC50 | = | 28.9 | uM | ALA4413422 | nM | Rattus norvegicus | |||
4. | ALA166 | melarsoprol | IC50 | = | 0.009 | uM | ALA4413418 | 8.06 | nM | Trypanosoma brucei rhodesiense | ||
5. | ALA166 | melarsoprol | IC50 | = | 0.02 | uM | ALA4411707 | 7.70 | nM | Trypanosoma brucei rhodesiense | ||
6. | ALA166 | melarsoprol | IC50 | = | 0.04 | uM | ALA4385220 | 7.40 | nM | Trypanosoma brucei rhodesiense | ||
7. | ALA166 | melarsoprol | IC50 | = | 0.04 | ug ml-1 | ALA4376350 | ug.mL-1 | Trypanosoma brucei rhodesiense | |||
8. | ALA166 | melarsoprol | IC50 | = | 0.2 | ug ml-1 | ALA4376349 | ug.mL-1 | Leishmania donovani | |||
9. | ALA166 | melarsoprol | IC50 | = | 0.001 | ug ml-1 | ALA4376346 | ug.mL-1 | Trypanosoma brucei rhodesiense | |||
10. | ALA166 | melarsoprol | IC50 | = | 5.42 | ug ml-1 | ALA4376347 | ug.mL-1 | Trypanosoma cruzi | |||
11. | ALA166 | melarsoprol | IC50 | = | 33.26 | ug ml-1 | ALA4376348 | ug.mL-1 | Leishmania donovani | |||
12. | ALA166 | melarsoprol | IC50 | = | 0.36 | ug ml-1 | ALA4376345 | ug.mL-1 | Trypanosoma cruzi | |||
13. | ALA166 | melarsoprol | pIC50 | = | 8.22 | ALA4775072 | 8.22 | nM | Trypanosoma brucei rhodesiense | |||
14. | ALA166 | melarsoprol | IC50 | = | 0.006 | uM | ALA4775072 | 8.22 | nM | Trypanosoma brucei rhodesiense | ||
15. | ALA166 | melarsoprol | IC50 | = | 7.78 | uM | ALA4734226 | 5.11 | nM | Rattus norvegicus | ||
16. | ALA166 | melarsoprol | Ratio IC50 | = | 1995 | ALA4734225 | ||||||
17. | ALA166 | melarsoprol | IC50 | = | 0.004 | uM | ALA4734224 | 8.41 | nM | Trypanosoma brucei rhodesiense | ||
18. | ALA166 | melarsoprol | IC50 | = | 0.011 | uM | ALA4733628 | 7.96 | nM | Trypanosoma brucei rhodesiense | ||
19. | ALA166 | melarsoprol | IC50 | = | 0.009 | uM | ALA4718738 | 8.05 | nM | Trypanosoma brucei rhodesiense | ||
20. | ALA166 | melarsoprol | IC50 | = | 0.007 | uM | ALA4343682 | 8.15 | nM | Trypanosoma brucei rhodesiense |