| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA74141 | 4 | Ki | = | 0.51 | nM | ALA5247025 | 9.29 | nM | Homo sapiens | ||
| 2. | ALA74141 | 4 | Selectivity | = | 125 | ALA745693 | Homo sapiens | |||||
| 3. | ALA74141 | 4 | AUC | = | 603 | ng hr ml-1 | ALA638329 | ng.hr.mL-1 | Rattus norvegicus | |||
| 4. | ALA74141 | 4 | clogP | = | 5 | ALA646685 | ||||||
| 5. | ALA74141 | 4 | PAR | = | 0.1 | mg kg-1 | ALA793163 | mg kg-1 | Rattus norvegicus | |||
| 6. | ALA74141 | 4 | Activity | = | 180 | % | ALA772851 | % | Rattus norvegicus | |||
| 7. | ALA74141 | 4 | Ki | = | 0.51 | nM | ALA748895 | 9.29 | nM | Homo sapiens | ||
| 8. | ALA74141 | 4 | AUC | = | 743 | ng hr ml-1 | ALA618582 | ng.hr.mL-1 | ||||
| 9. | ALA74141 | 4 | clogP | = | 4.3 | ALA625052 | ||||||
| 10. | ALA74141 | 4 | MD | = | 180 | % | ALA788181 | % | Rattus norvegicus | |||
| 11. | ALA74141 | 4 | AUC | = | 603 | ng hr ml-1 | ALA626550 | ng.hr.mL-1 | Rattus norvegicus | |||
| 12. | ALA74141 | 4 | Activity | = | 76 | % | ALA618983 | % | ||||
| 13. | ALA74141 | 4 | Selectivity ratio | = | 102.7 | ALA745726 | Homo sapiens | |||||
| 14. | ALA74141 | 4 | Selectivity ratio | = | 124.9 | ALA745725 | Homo sapiens | |||||
| 15. | ALA74141 | 4 | Ki | = | 0.51 | nM | ALA745193 | 9.29 | nM | Homo sapiens | ||
| 16. | ALA74141 | 4 | F | = | 9 | % | ALA620951 | % | ||||
| 17. | ALA74141 | 4 | F | = | 44 | % | ALA623068 | % | Rattus norvegicus | |||
| 18. | ALA74141 | 4 | cLogP | = | 5 | ALA883126 | ||||||
| 19. | ALA74141 | 4 | Acetylcholine release | = | 180 | % | ALA773475 | % | Rattus norvegicus | |||
| 20. | ALA74141 | 4 | AUC | = | 603 | ng hr ml-1 | ALA621609 | ng.hr.mL-1 |
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