| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA77131 | 24 | CLint | 64.57 | microL/min/1E6 cells | ALA3301372 | uL.min-1.(10^6cells)-1 | |||||
| 2. | ALA77131 | 24 | CLint | 33.88 | microL/min/1E6 cells | ALA3301371 | uL.min-1.(10^6cells)-1 | |||||
| 3. | ALA77131 | 24 | Fm | = | 0.55 | ALA3532079 | Homo sapiens | |||||
| 4. | ALA77131 | 24 | Fm | = | 0.49 | ALA3532078 | Homo sapiens | |||||
| 5. | ALA77131 | 24 | t1/2 | = | 3.2 | hr | ALA3539876 | hr | Rattus norvegicus | |||
| 6. | ALA77131 | 24 | Cmax | = | 1150 | ng/ml | ALA3539875 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 7. | ALA77131 | 24 | CLH | = | 17 | ml/min.kg | ALA3541915 | mL.min-1.kg-1 | Homo sapiens | |||
| 8. | ALA77131 | 24 | CL | = | 38 | ml/min.kg | ALA3541916 | mL.min-1.kg-1 | Homo sapiens | |||
| 9. | ALA77131 | 24 | F | < | 5 | % | ALA3541917 | % | Homo sapiens | |||
| 10. | ALA77131 | 24 | Retention_time | = | 10.9 | min | ALA3541918 | min | Homo sapiens | |||
| 11. | ALA77131 | 24 | AUC | = | 1630 | ng.hr/ml | ALA3539874 | ng.hr.mL-1 | Rattus norvegicus | |||
| 12. | ALA77131 | 24 | t1/2 | = | 1 | hr | ALA3539873 | hr | Cavia porcellus | |||
| 13. | ALA77131 | 24 | Cmax | = | 9.8 | ng/ml | ALA3539872 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Cavia porcellus | ||
| 14. | ALA77131 | 24 | AUC | = | 4.25 | ng.hr/ml | ALA3539871 | ng.hr.mL-1 | Cavia porcellus | |||
| 15. | ALA77131 | 24 | t1/2 | = | 0.5 | hr | ALA3539866 | hr | Rattus norvegicus | |||
| 16. | ALA77131 | 24 | AUC | = | 509 | ng.hr/ml | ALA3539865 | ng.hr.mL-1 | Rattus norvegicus | |||
| 17. | ALA77131 | 24 | t1/2 | = | 3.1 | hr | ALA3539864 | hr | Cavia porcellus | |||
| 18. | ALA77131 | 24 | AUC | = | 35.6 | ng.hr/ml | ALA3539863 | ng.hr.mL-1 | Cavia porcellus | |||
| 19. | ALA77131 | 24 | Drug metabolism | 0 | ALA3539885 | metabolite_detected | ||||||
| 20. | ALA77131 | 24 | Drug metabolism | 0 | ALA3539884 | metabolite_detected |
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