# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1908842 | 23, JNJ-28312141 | Kd | = | 310 | nM | ALA5252280 | 6.51 | nM | Homo sapiens | ||
2. | ALA1908842 | 23, JNJ-28312141 | Kd | = | 240 | nM | ALA5152919 | 6.62 | nM | Homo sapiens | ||
3. | ALA1908842 | 23, JNJ-28312141 | Kd | = | 2000 | nM | ALA4739795 | 5.70 | nM | Homo sapiens | ||
4. | ALA1908842 | 23, JNJ-28312141 | pKd | = | 5.7 | ALA4739795 | 5.70 | nM | Homo sapiens | |||
5. | ALA1908842 | 23, JNJ-28312141 | IC50 | = | 1.7 | nM | ALA5106447 | 8.77 | nM | |||
6. | ALA1908842 | 23, JNJ-28312141 | IC50 | = | 1.7 | nM | ALA5106387 | 8.77 | nM | |||
7. | ALA1908842 | 23, JNJ-28312141 | INH | = | 79 | % | ALA2161582 | % | Mus musculus | |||
8. | ALA1908842 | 23, JNJ-28312141 | INH | = | 65 | % | ALA2161581 | % | Mus musculus | |||
9. | ALA1908842 | 23, JNJ-28312141 | INH | = | 79 | % | ALA2161580 | % | Mus musculus | |||
10. | ALA1908842 | 23, JNJ-28312141 | Activity | = | 9.3 | mm | ALA2160237 | mm | Rattus norvegicus | |||
11. | ALA1908842 | 23, JNJ-28312141 | INH | 0 | ALA2162236 | Dose-dependent effect | % | Rattus norvegicus | ||||
12. | ALA1908842 | 23, JNJ-28312141 | Stability | = | 81 | % | ALA2160238 | % | Mus musculus | |||
13. | ALA1908842 | 23, JNJ-28312141 | INH | = | 74 | % | ALA2162250 | % | Rattus norvegicus | |||
14. | ALA1908842 | 23, JNJ-28312141 | INH | = | 100 | % | ALA2162249 | % | Rattus norvegicus | |||
15. | ALA1908842 | 23, JNJ-28312141 | INH | = | 100 | % | ALA2162248 | % | Rattus norvegicus | |||
16. | ALA1908842 | 23, JNJ-28312141 | INH | = | 40 | % | ALA2162246 | % | Rattus norvegicus | |||
17. | ALA1908842 | 23, JNJ-28312141 | INH | = | 66 | % | ALA2162245 | % | Rattus norvegicus | |||
18. | ALA1908842 | 23, JNJ-28312141 | INH | = | 97 | % | ALA2162244 | % | Rattus norvegicus | |||
19. | ALA1908842 | 23, JNJ-28312141 | INH | = | 34 | % | ALA2162242 | % | Rattus norvegicus | |||
20. | ALA1908842 | 23, JNJ-28312141 | INH | = | 43 | % | ALA2162241 | % | Rattus norvegicus |