| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1915863 | 10c | CL | = | 1.8 | ml/min.kg | ALA1918184 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 2. | ALA1915863 | 10c | F | = | 87 | % | ALA1918291 | % | Rattus norvegicus | |||
| 3. | ALA1915863 | 10c | Vdss | = | 669 | ml/kg | ALA1918290 | L.kg-1 | Rattus norvegicus | |||
| 4. | ALA1915863 | 10c | t1/2 | = | 5.6 | hr | ALA1918289 | hr | Rattus norvegicus | |||
| 5. | ALA1915863 | 10c | t1/2 | = | 6.5 | hr | ALA1918288 | hr | Rattus norvegicus | |||
| 6. | ALA1915863 | 10c | Cmax | = | 1.67 | ug ml-1 | ALA1918183 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 7. | ALA1915863 | 10c | AUC | = | 9.52 | microg.hr/mL | ALA1918181 | ng.hr.mL-1 | Rattus norvegicus | |||
| 8. | ALA1915863 | 10c | AUC | = | 8.28 | microg.hr/mL | ALA1918180 | ng.hr.mL-1 | Rattus norvegicus | |||
| 9. | ALA1915863 | 10c | INH | = | 58 | % | ALA1918139 | % | Cavia porcellus | |||
| 10. | ALA1915863 | 10c | Kinetic_solubility | = | 490 | ug ml-1 | ALA1918138 | ug.mL-1 | ||||
| 11. | ALA1915863 | 10c | IC50 | = | 8.1 | nM | ALA1918137 | 8.09 | nM | Homo sapiens | ||
| 12. | ALA1915863 | 10c | IC50 | = | 0.7 | nM | ALA1918136 | 9.15 | nM | Mus musculus | ||
| 13. | ALA1915863 | 10c | Ki | > | 10000 | nM | ALA1918135 | nM | Homo sapiens |
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