| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1922212 | alphaS-25 | IC50 | = | 35000 | nM | ALA3707632 | 4.46 | 267730 | nM | Homo sapiens | |
| 2. | ALA1922212 | alphaS-25 | IC50 | = | 70 | nM | ALA3705418 | 7.16 | 267680 | nM | Homo sapiens | |
| 3. | ALA1922212 | alphaS-25 | IC50 | > | 200000 | nM | ALA3707736 | 267720 | nM | Homo sapiens | ||
| 4. | ALA1922212 | alphaS-25 | IC50 | = | 12000 | nM | ALA3707784 | 4.92 | 267700 | nM | Homo sapiens | |
| 5. | ALA1922212 | alphaS-25 | F | = | 15 | % | ALA1926143 | % | Mus musculus | |||
| 6. | ALA1922212 | alphaS-25 | Ratio | = | 2 | ALA1926142 | Mus musculus | |||||
| 7. | ALA1922212 | alphaS-25 | CL | = | 0.024 | L/hr | ALA1926141 | L/hr | Mus musculus | |||
| 8. | ALA1922212 | alphaS-25 | Vd | = | 0.012 | l | ALA1926140 | l | Mus musculus | |||
| 9. | ALA1922212 | alphaS-25 | t1/2 | = | 0.4 | hr | ALA1926139 | hr | Mus musculus | |||
| 10. | ALA1922212 | alphaS-25 | AUC | = | 109.4 | micromol.hr/L | ALA1926138 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 11. | ALA1922212 | alphaS-25 | Cmax | = | 214.7 | umol/L | ALA1926137 | nM | Mus musculus | |||
| 12. | ALA1922212 | alphaS-25 | solubility | 0 | ALA1926136 | soluble | ||||||
| 13. | ALA1922212 | alphaS-25 | IC50 | = | 0.16 | uM | ALA1926135 | 6.80 | nM | Homo sapiens | ||
| 14. | ALA1922212 | alphaS-25 | Activity | = | 22 | % | ALA1926133 | % | Mus musculus | |||
| 15. | ALA1922212 | alphaS-25 | Ratio IC50 | = | 60 | ALA1926132 | ||||||
| 16. | ALA1922212 | alphaS-25 | Ratio IC50 | = | 80 | ALA1926131 | ||||||
| 17. | ALA1922212 | alphaS-25 | GI50 | = | 5.4 | uM | ALA1926130 | nM | Homo sapiens | |||
| 18. | ALA1922212 | alphaS-25 | GI50 | = | 5.4 | uM | ALA1926129 | nM | Homo sapiens | |||
| 19. | ALA1922212 | alphaS-25 | GI50 | = | 4.1 | uM | ALA1926128 | nM | Homo sapiens | |||
| 20. | ALA1922212 | alphaS-25 | GI50 | = | 6.8 | uM | ALA1926127 | nM | Homo sapiens |
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