# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1922219 | alphaSbetaR-21, CCT68127 | IC50 | = | 520 | nM | ALA5224416 | 6.28 | nM | Homo sapiens | ||
2. | ALA1922219 | alphaSbetaR-21, CCT68127 | IC50 | = | 70 | nM | ALA5224415 | 7.16 | nM | Homo sapiens | ||
3. | ALA1922219 | alphaSbetaR-21, CCT68127 | IC50 | = | 4800 | nM | ALA5224414 | 5.32 | nM | Homo sapiens | ||
4. | ALA1922219 | alphaSbetaR-21, CCT68127 | IC50 | = | 110 | nM | ALA5224413 | 6.96 | nM | Homo sapiens | ||
5. | ALA1922219 | alphaSbetaR-21, CCT68127 | IC50 | = | 1100 | nM | ALA5224412 | 5.96 | nM | Homo sapiens | ||
6. | ALA1922219 | alphaSbetaR-21, CCT68127 | IC50 | = | 90 | nM | ALA5224411 | 7.05 | nM | Homo sapiens | ||
7. | ALA1922219 | alphaSbetaR-21, CCT68127 | IC50 | = | 6200 | nM | ALA5224410 | 5.21 | nM | Homo sapiens | ||
8. | ALA1922219 | alphaSbetaR-21, CCT68127 | Activity | 0 | ALA1926218 | Active | Homo sapiens | |||||
9. | ALA1922219 | alphaSbetaR-21, CCT68127 | Activity | 0 | ALA1926150 | Active | Homo sapiens | |||||
10. | ALA1922219 | alphaSbetaR-21, CCT68127 | IC50 | = | 107 | nM | ALA1926149 | 6.97 | nM | Homo sapiens | ||
11. | ALA1922219 | alphaSbetaR-21, CCT68127 | IC50 | = | 1.3 | uM | ALA1926148 | 5.89 | nM | Homo sapiens | ||
12. | ALA1922219 | alphaSbetaR-21, CCT68127 | Activity | 0 | ALA1926147 | Active | Homo sapiens | |||||
13. | ALA1922219 | alphaSbetaR-21, CCT68127 | INH | 0 | ALA1926146 | Active | % | Homo sapiens | ||||
14. | ALA1922219 | alphaSbetaR-21, CCT68127 | Activity | 0 | ALA1926145 | Active | Homo sapiens | |||||
15. | ALA1922219 | alphaSbetaR-21, CCT68127 | Activity | = | 49 | % | ALA1926144 | % | Homo sapiens | |||
16. | ALA1922219 | alphaSbetaR-21, CCT68127 | F | = | 15 | % | ALA1926143 | % | Mus musculus | |||
17. | ALA1922219 | alphaSbetaR-21, CCT68127 | Ratio | = | 2 | ALA1926142 | Mus musculus | |||||
18. | ALA1922219 | alphaSbetaR-21, CCT68127 | CL | = | 0.009 | L/hr | ALA1926141 | L/hr | Mus musculus | |||
19. | ALA1922219 | alphaSbetaR-21, CCT68127 | Vd | = | 0.013 | l | ALA1926140 | l | Mus musculus | |||
20. | ALA1922219 | alphaSbetaR-21, CCT68127 | t1/2 | = | 2.8 | hr | ALA1926139 | hr | Mus musculus |