| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1927157 | 7m | CL | = | 1.02 | L/kg/hr | ALA1931597 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 2. | ALA1927157 | 7m | t1/2 | = | 3.63 | hr | ALA1931596 | hr | Rattus norvegicus | |||
| 3. | ALA1927157 | 7m | Tmax | = | 0.25 | hr | ALA1931595 | hr | Rattus norvegicus | |||
| 4. | ALA1927157 | 7m | Cmax | = | 11298 | ng/ml | ALA1931594 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 5. | ALA1927157 | 7m | F | = | 42 | % | ALA1931593 | % | Rattus norvegicus | |||
| 6. | ALA1927157 | 7m | AUC | = | 9901 | hr.ng/ml | ALA1931592 | ng.hr.mL-1 | Rattus norvegicus | |||
| 7. | ALA1927157 | 7m | Vdss | = | 0.47 | L/Kg | ALA1931591 | L.kg-1 | Rattus norvegicus | |||
| 8. | ALA1927157 | 7m | CL | = | 0.46 | L/kg/hr | ALA1931509 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 9. | ALA1927157 | 7m | t1/2 | = | 5.62 | hr | ALA1931508 | hr | Rattus norvegicus | |||
| 10. | ALA1927157 | 7m | Cmax | = | 21827 | ng/ml | ALA1931507 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 11. | ALA1927157 | 7m | AUC | = | 11819 | hr.ng/ml | ALA1931506 | ng.hr.mL-1 | Rattus norvegicus | |||
| 12. | ALA1927157 | 7m | Fu | = | 2.6 | % | ALA1932801 | Rattus norvegicus | ||||
| 13. | ALA1927157 | 7m | logD | = | 1.1 | ALA1932800 | ||||||
| 14. | ALA1927157 | 7m | Ratio | = | 10.1 | ALA1932799 | Homo sapiens | |||||
| 15. | ALA1927157 | 7m | Papp | = | 1.8 | 10'-6 cm/s | ALA1932798 | 10'-6 cm/s | Homo sapiens | |||
| 16. | ALA1927157 | 7m | CLH | = | 27.5 | uL/min | ALA1932797 | uL/min | Rattus norvegicus | |||
| 17. | ALA1927157 | 7m | CLH | = | 13.9 | uL/min | ALA1932796 | uL/min | Homo sapiens | |||
| 18. | ALA1927157 | 7m | Ki | = | 543 | nM | ALA1931065 | 6.26 | nM | Homo sapiens | ||
| 19. | ALA1927157 | 7m | Ki | = | 67 | nM | ALA1931064 | 7.17 | nM | Homo sapiens | ||
| 20. | ALA1927157 | 7m | Ki | = | 1140 | nM | ALA1931063 | 5.94 | nM | Homo sapiens |
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