| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1935538 | 10, CSUOH0901, NSC751382 | Ratio IC50 | = | 0.1 | ALA2072970 | ||||||
| 2. | ALA1935538 | 10, CSUOH0901, NSC751382 | IC50 | = | 3.22 | uM | ALA2072968 | 5.49 | nM | Trypanosoma brucei | ||
| 3. | ALA1935538 | 10, CSUOH0901, NSC751382 | IC50 | = | 0.39 | uM | ALA2339661 | 6.41 | nM | Homo sapiens | ||
| 4. | ALA1935538 | 10, CSUOH0901, NSC751382 | IC50 | = | 0.77 | uM | ALA2339660 | 6.11 | nM | Homo sapiens | ||
| 5. | ALA1935538 | 10, CSUOH0901, NSC751382 | Ratio IC50 | = | 1.7 | ALA2339659 | Homo sapiens | |||||
| 6. | ALA1935538 | 10, CSUOH0901, NSC751382 | INH | > | 90 | % | ALA2339658 | % | Homo sapiens | |||
| 7. | ALA1935538 | 10, CSUOH0901, NSC751382 | INH | 0 | ALA2060035 | Active | % | Homo sapiens | ||||
| 8. | ALA1935538 | 10, CSUOH0901, NSC751382 | INH | 0 | ALA2060034 | Active | % | Homo sapiens | ||||
| 9. | ALA1935538 | 10, CSUOH0901, NSC751382 | Activity | 0 | ALA2060030 | Active | Homo sapiens | |||||
| 10. | ALA1935538 | 10, CSUOH0901, NSC751382 | INH | 0 | ALA2060029 | Active | % | Homo sapiens | ||||
| 11. | ALA1935538 | 10, CSUOH0901, NSC751382 | INH | 0 | ALA2060028 | Active | % | Homo sapiens | ||||
| 12. | ALA1935538 | 10, CSUOH0901, NSC751382 | INH | 0 | ALA2060026 | Dose-dependent effect | % | |||||
| 13. | ALA1935538 | 10, CSUOH0901, NSC751382 | IC50 | = | 0.2 | uM | ALA3587752 | 6.70 | nM | Homo sapiens | ||
| 14. | ALA1935538 | 10, CSUOH0901, NSC751382 | Tmax | = | 2 | hr | ALA1938035 | hr | Rattus norvegicus | |||
| 15. | ALA1935538 | 10, CSUOH0901, NSC751382 | Ratio IC50 | = | 10 | ALA1938043 | Homo sapiens | |||||
| 16. | ALA1935538 | 10, CSUOH0901, NSC751382 | Ratio IC50 | = | 1000 | ALA1938042 | Homo sapiens | |||||
| 17. | ALA1935538 | 10, CSUOH0901, NSC751382 | MRT | = | 6 | hr | ALA1938040 | hr | Rattus norvegicus | |||
| 18. | ALA1935538 | 10, CSUOH0901, NSC751382 | CL/F | = | 0.48 | L/hr | ALA1938039 | L/hr | Rattus norvegicus | |||
| 19. | ALA1935538 | 10, CSUOH0901, NSC751382 | IC50 | = | 0.2 | uM | ALA1937551 | 6.70 | nM | Homo sapiens | ||
| 20. | ALA1935538 | 10, CSUOH0901, NSC751382 | Activity | = | 3.12 | % | ALA1937550 | % | Homo sapiens |
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