| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1939559 | 25 | CL | = | 0.49 | ml/hr.kg | ALA5257211 | mL.min-1.kg-1 | ||||
| 2. | ALA1939559 | 25 | t1/2 | = | 4 | hr | ALA5257210 | hr | ||||
| 3. | ALA1939559 | 25 | F | = | 69 | % | ALA5257209 | % | ||||
| 4. | ALA1939559 | 25 | pIC50 | = | 8.3 | ALA5257208 | 8.30 | nM | Homo sapiens | |||
| 5. | ALA1939559 | 25 | pIC50 | = | 8.2 | ALA5257202 | 8.20 | nM | Homo sapiens | |||
| 6. | ALA1939559 | 25 | IC50 | > | 10 | uM | ALA1941432 | nM | Homo sapiens | |||
| 7. | ALA1939559 | 25 | Drug uptake | = | 3.4 | mg kg-1 | ALA1941431 | mg kg-1 | Mus musculus | |||
| 8. | ALA1939559 | 25 | Drug uptake | = | 1.3 | mg kg-1 | ALA1941430 | mg kg-1 | Mus musculus | |||
| 9. | ALA1939559 | 25 | Drug uptake | = | 5.6 | mg kg-1 | ALA1941429 | mg kg-1 | Mus musculus | |||
| 10. | ALA1939559 | 25 | EC | = | 1 | mg kg-1 | ALA1941428 | mg kg-1 | Mus musculus | |||
| 11. | ALA1939559 | 25 | IC50 | = | 200 | nM | ALA1941427 | 6.70 | nM | Mus musculus | ||
| 12. | ALA1939559 | 25 | IC50 | = | 9.8 | nM | ALA1941426 | 8.01 | nM | Homo sapiens | ||
| 13. | ALA1939559 | 25 | t1/2 | = | 9 | hr | ALA1941425 | hr | Macaca fascicularis | |||
| 14. | ALA1939559 | 25 | t1/2 | = | 1 | hr | ALA1941424 | hr | Canis lupus familiaris | |||
| 15. | ALA1939559 | 25 | t1/2 | = | 4 | hr | ALA1941423 | hr | Rattus norvegicus | |||
| 16. | ALA1939559 | 25 | t1/2 | = | 4 | hr | ALA1941422 | hr | Mus musculus | |||
| 17. | ALA1939559 | 25 | Fu | = | 3.7 | % | ALA1941421 | Macaca fascicularis | ||||
| 18. | ALA1939559 | 25 | Fu | = | 1.5 | % | ALA1941420 | Canis lupus familiaris | ||||
| 19. | ALA1939559 | 25 | Fu | = | 6.1 | % | ALA1941419 | Rattus norvegicus | ||||
| 20. | ALA1939559 | 25 | Fu | = | 0.7 | % | ALA1941418 | Mus musculus |
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