# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1940404 | 7 | Ki | = | 2228 | nM | ALA3366168 | 5.65 | nM | Homo sapiens | ||
2. | ALA1940404 | 7 | Ki | = | 3959 | nM | ALA3366167 | 5.40 | nM | Homo sapiens | ||
3. | ALA1940404 | 7 | Ki | > | 10000 | nM | ALA3366166 | nM | Homo sapiens | |||
4. | ALA1940404 | 7 | Ki | = | 698.6 | nM | ALA3366162 | 6.16 | nM | Homo sapiens | ||
5. | ALA1940404 | 7 | Ki | > | 10000 | nM | ALA3366161 | nM | Rattus norvegicus | |||
6. | ALA1940404 | 7 | Ki | = | 1622 | nM | ALA3366160 | 5.79 | nM | Homo sapiens | ||
7. | ALA1940404 | 7 | Ki | = | 103 | nM | ALA3366159 | 6.99 | nM | Homo sapiens | ||
8. | ALA1940404 | 7 | Ki | = | 4.3 | nM | ALA3366158 | 8.37 | nM | Rattus norvegicus | ||
9. | ALA1940404 | 7 | Ki | = | 49 | nM | ALA3366157 | 7.31 | nM | Homo sapiens | ||
10. | ALA1940404 | 7 | Ki | = | 8.8 | nM | ALA3366156 | 8.06 | nM | Homo sapiens | ||
11. | ALA1940404 | 7 | Ki | = | 22 | nM | ALA3366155 | 7.66 | nM | Homo sapiens | ||
12. | ALA1940404 | 7 | Ki | = | 656 | nM | ALA3366154 | 6.18 | nM | Homo sapiens | ||
13. | ALA1940404 | 7 | Ki | = | 72 | nM | ALA3366153 | 7.14 | nM | Homo sapiens | ||
14. | ALA1940404 | 7 | Ki | = | 317 | nM | ALA3366152 | 6.50 | nM | Homo sapiens | ||
15. | ALA1940404 | 7 | pKi | = | 8.97 | ALA4416273 | 8.97 | nM | Homo sapiens | |||
16. | ALA1940404 | 7 | pKd | = | 9.1 | ALA4416273 | 9.10 | nM | Homo sapiens | |||
17. | ALA1940404 | 7 | t1/2 | = | 0.81 | min | ALA4416272 | hr | Homo sapiens | |||
18. | ALA1940404 | 7 | Kdiss | = | 0.91 | /min | ALA4416271 | /min | Homo sapiens | |||
19. | ALA1940404 | 7 | Ka | = | 1.22 | 10'9/M/min | ALA4416270 | 10'9/M/min | Homo sapiens | |||
20. | ALA1940404 | 7 | Activity | 0 | ALA4416278 | Active | Homo sapiens |