# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1944785 | [18F]12a, [18F]GE-180 | Ki | = | 2.4 | nM | ALA5228258 | 8.62 | nM | Homo sapiens | ||
2. | ALA1944785 | [18F]12a, [18F]GE-180 | Activity | = | 64 | % | ALA1948440 | % | Rattus norvegicus | |||
3. | ALA1944785 | [18F]12a, [18F]GE-180 | Activity | = | 64 | % | ALA1948450 | % | Rattus norvegicus | |||
4. | ALA1944785 | [18F]12a, [18F]GE-180 | Activity | = | 86 | % | ALA1948439 | % | Rattus norvegicus | |||
5. | ALA1944785 | [18F]12a, [18F]GE-180 | Activity | = | 86 | % | ALA1948449 | % | Rattus norvegicus | |||
6. | ALA1944785 | [18F]12a, [18F]GE-180 | Stability | = | 94 | % | ALA1948447 | % | Rattus norvegicus | |||
7. | ALA1944785 | [18F]12a, [18F]GE-180 | Ratio | = | 3.07 | ALA1948446 | ||||||
8. | ALA1944785 | [18F]12a, [18F]GE-180 | Ratio | = | 3.21 | ALA1948445 | ||||||
9. | ALA1944785 | [18F]12a, [18F]GE-180 | Drug uptake | = | 0.45 | % ID/g | ALA1948444 | % ID/g | Rattus norvegicus | |||
10. | ALA1944785 | [18F]12a, [18F]GE-180 | Drug uptake | = | 0.53 | % ID/g | ALA1948443 | % ID/g | Rattus norvegicus | |||
11. | ALA1944785 | [18F]12a, [18F]GE-180 | Ki | = | 0.87 | nM | ALA1948441 | 9.06 | nM | Rattus norvegicus |