# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1949930 | 15k, enantiomer 1 | F | = | 11 | % | ALA1953620 | % | Rattus norvegicus | |||
2. | ALA1949930 | 15k, enantiomer 1 | Activity | 0 | ALA1953619 | Dose-dependent effect | Rattus norvegicus | |||||
3. | ALA1949930 | 15k, enantiomer 1 | Activity | = | 35 | % | ALA1953618 | % | Rattus norvegicus | |||
4. | ALA1949930 | 15k, enantiomer 1 | Activity | = | 21 | % | ALA1953617 | % | Rattus norvegicus | |||
5. | ALA1949930 | 15k, enantiomer 1 | Activity | = | 22 | % | ALA1953616 | % | Rattus norvegicus | |||
6. | ALA1949930 | 15k, enantiomer 1 | IC50 | = | 9.54 | mg kg-1 | ALA1953615 | mg kg-1 | Rattus norvegicus | |||
7. | ALA1949930 | 15k, enantiomer 1 | INH | 0 | ALA1953615 | Dose-dependent effect | % | Rattus norvegicus | ||||
8. | ALA1949930 | 15k, enantiomer 1 | IC50 | = | 3.9 | uM | ALA1953198 | 5.41 | nM | |||
9. | ALA1949930 | 15k, enantiomer 1 | IC50 | = | 4.4 | uM | ALA1953197 | 5.36 | nM | Homo sapiens | ||
10. | ALA1949930 | 15k, enantiomer 1 | IC50 | = | 6.3 | uM | ALA1953196 | 5.20 | nM | Homo sapiens | ||
11. | ALA1949930 | 15k, enantiomer 1 | IC50 | = | 4.8 | uM | ALA1953195 | 5.32 | nM | Homo sapiens | ||
12. | ALA1949930 | 15k, enantiomer 1 | IC50 | = | 7.9 | uM | ALA1953194 | 5.10 | nM | Homo sapiens | ||
13. | ALA1949930 | 15k, enantiomer 1 | IC50 | = | 2.2 | uM | ALA1953193 | 5.66 | nM | Homo sapiens | ||
14. | ALA1949930 | 15k, enantiomer 1 | INH | > | 50 | % | ALA1953192 | % | ||||
15. | ALA1949930 | 15k, enantiomer 1 | INH | > | 50 | % | ALA1953191 | % | Homo sapiens | |||
16. | ALA1949930 | 15k, enantiomer 1 | INH | > | 50 | % | ALA1953190 | % | Homo sapiens | |||
17. | ALA1949930 | 15k, enantiomer 1 | INH | > | 50 | % | ALA1953189 | % | Homo sapiens | |||
18. | ALA1949930 | 15k, enantiomer 1 | INH | > | 50 | % | ALA1953188 | % | Homo sapiens | |||
19. | ALA1949930 | 15k, enantiomer 1 | INH | > | 50 | % | ALA1953187 | % | Homo sapiens | |||
20. | ALA1949930 | 15k, enantiomer 1 | IC50 | = | 3.3 | uM | ALA1953186 | 5.48 | nM | Homo sapiens |