# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1950743 | 17b | IC50 | = | 21 | uM | ALA1952486 | 4.68 | nM | Homo sapiens | ||
2. | ALA1950743 | 17b | Activity | 0 | ALA1952517 | Not Active | Rattus norvegicus | |||||
3. | ALA1950743 | 17b | Activity | 0 | ALA1952516 | Active | Rattus norvegicus | |||||
4. | ALA1950743 | 17b | Time | = | 196 | min | ALA1952515 | hr | Rattus norvegicus | |||
5. | ALA1950743 | 17b | Activity | = | 98 | % | ALA1952514 | % | Rattus norvegicus | |||
6. | ALA1950743 | 17b | Activity | = | 84 | % | ALA1952513 | % | Rattus norvegicus | |||
7. | ALA1950743 | 17b | Activity | = | 193 | % | ALA1952512 | % | Rattus norvegicus | |||
8. | ALA1950743 | 17b | Activity | = | 152 | % | ALA1952511 | % | Rattus norvegicus | |||
9. | ALA1950743 | 17b | Activity | = | 90 | % | ALA1952510 | % | Rattus norvegicus | |||
10. | ALA1950743 | 17b | Time | = | 116 | min | ALA1952509 | hr | Rattus norvegicus | |||
11. | ALA1950743 | 17b | Time | = | 122 | min | ALA1952508 | hr | Rattus norvegicus | |||
12. | ALA1950743 | 17b | Time | = | 115 | min | ALA1952507 | hr | Rattus norvegicus | |||
13. | ALA1950743 | 17b | Activity | = | 45 | % | ALA1952506 | % | Rattus norvegicus | |||
14. | ALA1950743 | 17b | Activity | 0 | ALA1952505 | Dose-dependent effect | Rattus norvegicus | |||||
15. | ALA1950743 | 17b | INH | 0 | ALA1952504 | Dose-dependent effect | % | Rattus norvegicus | ||||
16. | ALA1950743 | 17b | ED50 | = | 0.14 | mg kg-1 | ALA1952504 | mg.kg-1 | Rattus norvegicus | |||
17. | ALA1950743 | 17b | PPB | = | 50 | % | ALA1952503 | % | Homo sapiens | |||
18. | ALA1950743 | 17b | PPB | = | 50 | % | ALA1952502 | % | Canis lupus familiaris | |||
19. | ALA1950743 | 17b | PPB | = | 50 | % | ALA1952501 | % | Rattus norvegicus | |||
20. | ALA1950743 | 17b | Selectivity ratio | > | 1000 | ALA1952500 |