| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1951346 | 36 | IC50 | = | 62 | nM | ALA5244639 | 7.21 | nM | Homo sapiens | ||
| 2. | ALA1951346 | 36 | F | = | 0 | % | ALA3411324 | % | Rattus norvegicus | |||
| 3. | ALA1951346 | 36 | Cmax | = | 8.5 | uM | ALA3411323 | nM | Rattus norvegicus | |||
| 4. | ALA1951346 | 36 | AUC | = | 4.3 | uM.hr | ALA3411322 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 5. | ALA1951346 | 36 | t1/2 | = | 1 | hr | ALA3411321 | hr | Rattus norvegicus | |||
| 6. | ALA1951346 | 36 | Vd | = | 0.3 | L/Kg | ALA3411320 | L.kg-1 | Rattus norvegicus | |||
| 7. | ALA1951346 | 36 | CL | = | 9 | ml/min.kg | ALA3411319 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 8. | ALA1951346 | 36 | IC50 | > | 1000 | nM | ALA3411315 | nM | Rattus norvegicus | |||
| 9. | ALA1951346 | 36 | t1/2 | = | 44 | min | ALA3411314 | hr | Rattus norvegicus | |||
| 10. | ALA1951346 | 36 | t1/2 | = | 33 | min | ALA3411313 | hr | Homo sapiens | |||
| 11. | ALA1951346 | 36 | INH | = | 34 | % | ALA3411306 | % | Homo sapiens | |||
| 12. | ALA1951346 | 36 | INH | = | 16 | % | ALA3411305 | % | Homo sapiens | |||
| 13. | ALA1951346 | 36 | INH | = | 49 | % | ALA3411304 | % | Homo sapiens | |||
| 14. | ALA1951346 | 36 | INH | = | 33 | % | ALA3411303 | % | Homo sapiens | |||
| 15. | ALA1951346 | 36 | IC50 | = | 7738 | nM | ALA3411302 | 5.11 | nM | Homo sapiens | ||
| 16. | ALA1951346 | 36 | IC50 | = | 1283 | nM | ALA3411301 | 5.89 | nM | Homo sapiens | ||
| 17. | ALA1951346 | 36 | Ratio IC50 | = | 26 | ALA3411300 | ||||||
| 18. | ALA1951346 | 36 | IC50 | = | 62 | nM | ALA3411298 | 7.21 | nM | Homo sapiens | ||
| 19. | ALA1951346 | 36 | IC50 | = | 1608 | nM | ALA3411299 | 5.79 | nM | Homo sapiens | ||
| 20. | ALA1951346 | 36 | Ratio IC50 | = | 3 | ALA1953086 |
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