# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1967116 | SID103904313 | GI | > | 70 | % | ALA2024790 | % | Homo sapiens | |||
2. | ALA1967116 | SID103904313 | F | = | 59 | % | ALA2024789 | % | Mus musculus | |||
3. | ALA1967116 | SID103904313 | AUC | = | 5.64 | microg.hr/mL | ALA2024788 | ng.hr.mL-1 | Mus musculus | |||
4. | ALA1967116 | SID103904313 | CL | = | 1.1 | L/hr.Kg | ALA2024787 | mL.min-1.kg-1 | Mus musculus | |||
5. | ALA1967116 | SID103904313 | Vd | = | 2.3 | L/Kg | ALA2024786 | L.kg-1 | Mus musculus | |||
6. | ALA1967116 | SID103904313 | t1/2 | = | 1.5 | hr | ALA2024785 | hr | Mus musculus | |||
7. | ALA1967116 | SID103904313 | EC15 | = | 55 | nM | ALA2024779 | nM | Homo sapiens | |||
8. | ALA1967116 | SID103904313 | IC50 | = | 14 | nM | ALA2024778 | 7.85 | nM | Homo sapiens | ||
9. | ALA1967116 | SID103904313 | IC50 | = | 16 | nM | ALA2024777 | 7.80 | nM | Homo sapiens | ||
10. | ALA1967116 | SID103904313 | IC50 | = | 3 | nM | ALA2024776 | 8.52 | nM | Homo sapiens | ||
11. | ALA1967116 | SID103904313 | ED50 | = | 1 | mg kg-1 | ALA2024780 | mg.kg-1 | Mus musculus | |||
12. | ALA1967116 | SID103904313 | pKi | < | 5.1 | ALA1963829 | inactive | nM | Homo sapiens | |||
13. | ALA1967116 | SID103904313 | pKi | = | 7.2 | ALA1963823 | 7.20 | active | nM | Homo sapiens | ||
14. | ALA1967116 | SID103904313 | pKi | = | 8.2 | ALA1963817 | 8.20 | active | nM | Homo sapiens | ||
15. | ALA1967116 | SID103904313 | pKi | < | 5.4 | ALA1963833 | inactive | nM | Homo sapiens | |||
16. | ALA1967116 | SID103904313 | pKi | = | 7.8 | ALA1963828 | 7.80 | active | nM | Homo sapiens | ||
17. | ALA1967116 | SID103904313 | pKi | < | 5 | ALA1963822 | inactive | nM | Homo sapiens | |||
18. | ALA1967116 | SID103904313 | pKi | < | 8.6 | ALA1963810 | inactive | nM | Homo sapiens | |||
19. | ALA1967116 | SID103904313 | pKi | < | 5 | ALA1963837 | inactive | nM | Homo sapiens | |||
20. | ALA1967116 | SID103904313 | pKi | < | 5.2 | ALA1963816 | inactive | nM | Homo sapiens |