| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA81521 | 12 | Selectivity | = | 890 | ALA824716 | Homo sapiens | |||||
| 2. | ALA81521 | 12 | F | = | 9 | % | ALA623340 | % | Canis lupus familiaris | |||
| 3. | ALA81521 | 12 | T1/2 | = | 1 | hr | ALA873810 | hr | Canis lupus familiaris | |||
| 4. | ALA81521 | 12 | T1/2 | = | 0.16 | hr | ALA618820 | hr | Canis lupus familiaris | |||
| 5. | ALA81521 | 12 | Volume | = | 0.53 | l kg-1 | ALA619814 | L.kg-1 | Canis lupus familiaris | |||
| 6. | ALA81521 | 12 | Clearance | = | 6.4 | ml min-1 kg-1 | ALA621389 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 7. | ALA81521 | 12 | F | = | 2 | % | ALA624106 | % | Rattus norvegicus | |||
| 8. | ALA81521 | 12 | T1/2 | = | 0.8 | hr | ALA624064 | hr | Rattus norvegicus | |||
| 9. | ALA81521 | 12 | T1/2 | = | 0.12 | hr | ALA624063 | hr | Rattus norvegicus | |||
| 10. | ALA81521 | 12 | Volume | = | 0.31 | l kg-1 | ALA627067 | L.kg-1 | Rattus norvegicus | |||
| 11. | ALA81521 | 12 | Clearance | = | 21.2 | ml min-1 kg-1 | ALA621093 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 12. | ALA81521 | 12 | Inhibition | = | 38.7 | % | ALA663031 | % | Homo sapiens | |||
| 13. | ALA81521 | 12 | Ki | = | 3.3 | nM | ALA847107 | 8.48 | nM | Bos taurus | ||
| 14. | ALA81521 | 12 | Ki | = | 4.97 | nM | ALA663260 | 8.30 | nM | Bos taurus | ||
| 15. | ALA81521 | 12 | Ki | = | 1930 | nM | ALA817823 | 5.71 | nM | Homo sapiens | ||
| 16. | ALA81521 | 12 | Ki | = | 2.17 | nM | ALA813625 | 8.66 | nM | Homo sapiens |
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