| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA82433 | 7 | Fold selectivity | = | 181 | ALA845306 | Homo sapiens | |||||
| 2. | ALA82433 | 7 | Fold selectivity | = | 57 | ALA844101 | Homo sapiens | |||||
| 3. | ALA82433 | 7 | Fold selectivity | = | 97 | ALA820226 | Homo sapiens | |||||
| 4. | ALA82433 | 7 | Fold selectivity | = | 1 | ALA845305 | Homo sapiens | |||||
| 5. | ALA82433 | 7 | Fold selectivity | = | 6 | ALA845304 | Homo sapiens | |||||
| 6. | ALA82433 | 7 | Fold selectivity | = | 11 | ALA845303 | Homo sapiens | |||||
| 7. | ALA82433 | 7 | F | 0 | % | ALA623175 | Not Determined | % | Canis lupus familiaris | |||
| 8. | ALA82433 | 7 | Vdss | = | 7.9 | l kg-1 | ALA624237 | L.kg-1 | Canis lupus familiaris | |||
| 9. | ALA82433 | 7 | CL | = | 8.9 | ml min-1 kg-1 | ALA624444 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 10. | ALA82433 | 7 | T1/2 | = | 10.4 | hr | ALA624301 | hr | Canis lupus familiaris | |||
| 11. | ALA82433 | 7 | F | = | 73 | % | ALA624101 | % | Rattus norvegicus | |||
| 12. | ALA82433 | 7 | Vdss | = | 3.9 | l kg-1 | ALA618537 | L.kg-1 | Rattus norvegicus | |||
| 13. | ALA82433 | 7 | CL | = | 17.3 | ml min-1 kg-1 | ALA623519 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 14. | ALA82433 | 7 | T1/2 | = | 2.9 | hr | ALA626924 | hr | Rattus norvegicus | |||
| 15. | ALA82433 | 7 | Solubility | = | 8.4 | mg ml-1 | ALA632908 | ug.mL-1 | ||||
| 16. | ALA82433 | 7 | Solubility | = | 33.9 | mg ml-1 | ALA632910 | ug.mL-1 | ||||
| 17. | ALA82433 | 7 | Binding | = | 80.7 | % | ALA766143 | % | ||||
| 18. | ALA82433 | 7 | logP | = | 2.25 | ALA630086 | ||||||
| 19. | ALA82433 | 7 | IC50 | = | 37 | nM | ALA690868 | 7.43 | nM | Homo sapiens | ||
| 20. | ALA82433 | 7 | IC50 | = | 25 | nM | ALA818933 | 7.60 | nM | Homo sapiens |
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