| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA83279 | 3 | Fold selectivity | = | 62 | ALA845306 | Homo sapiens | |||||
| 2. | ALA83279 | 3 | Fold selectivity | = | 47 | ALA844101 | Homo sapiens | |||||
| 3. | ALA83279 | 3 | Fold selectivity | = | 60 | ALA820226 | Homo sapiens | |||||
| 4. | ALA83279 | 3 | Fold selectivity | = | 0.5 | ALA845305 | Homo sapiens | |||||
| 5. | ALA83279 | 3 | Fold selectivity | = | 6 | ALA845304 | Homo sapiens | |||||
| 6. | ALA83279 | 3 | Fold selectivity | = | 5 | ALA845303 | Homo sapiens | |||||
| 7. | ALA83279 | 3 | F | 0 | % | ALA623174 | Not Determined | % | Canis lupus familiaris | |||
| 8. | ALA83279 | 3 | Vdss | = | 3.1 | l kg-1 | ALA624237 | L.kg-1 | Canis lupus familiaris | |||
| 9. | ALA83279 | 3 | CL | = | 4.6 | ml min-1 kg-1 | ALA624444 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 10. | ALA83279 | 3 | T1/2 | = | 5.2 | hr | ALA624301 | hr | Canis lupus familiaris | |||
| 11. | ALA83279 | 3 | F | = | 76 | % | ALA624100 | % | Rattus norvegicus | |||
| 12. | ALA83279 | 3 | Vdss | = | 1.9 | l kg-1 | ALA618536 | L.kg-1 | Rattus norvegicus | |||
| 13. | ALA83279 | 3 | CL | = | 14.4 | ml min-1 kg-1 | ALA622806 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 14. | ALA83279 | 3 | T1/2 | = | 6.1 | hr | ALA626923 | hr | Rattus norvegicus | |||
| 15. | ALA83279 | 3 | Solubility | < | 0 | mg ml-1 | ALA632908 | ug.mL-1 | ||||
| 16. | ALA83279 | 3 | Solubility | = | 0.12 | mg ml-1 | ALA632903 | ug.mL-1 | ||||
| 17. | ALA83279 | 3 | Binding | = | 99.4 | % | ALA766143 | % | ||||
| 18. | ALA83279 | 3 | logP | = | 4.29 | ALA630086 | ||||||
| 19. | ALA83279 | 3 | IC50 | = | 87 | nM | ALA690868 | 7.06 | nM | Homo sapiens | ||
| 20. | ALA83279 | 3 | IC50 | = | 14 | nM | ALA818933 | 7.85 | nM | Homo sapiens |
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