# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2012686 | 21 | Stability | 0 | ALA4370008 | Stable | % | |||||
2. | ALA2012686 | 21 | Activity | 0 | ALA4370009 | Toxic | ||||||
3. | ALA2012686 | 21 | Emax | = | 50 | % | ALA4370003 | % | Homo sapiens | |||
4. | ALA2012686 | 21 | EC50 | = | 1.37 | uM | ALA4370002 | 5.86 | nM | Homo sapiens | ||
5. | ALA2012686 | 21 | Emax | = | 119 | % | ALA4370001 | % | Rattus norvegicus | |||
6. | ALA2012686 | 21 | EC50 | = | 6.65 | nM | ALA4370000 | 8.18 | nM | Rattus norvegicus | ||
7. | ALA2012686 | 21 | Stability | 0 | ALA4370007 | Stable | % | |||||
8. | ALA2012686 | 21 | INH | = | 34 | % | ALA4369924 | % | Mus musculus | |||
9. | ALA2012686 | 21 | Activity | 0 | ALA4369979 | Non-Toxic | ||||||
10. | ALA2012686 | 21 | F | = | 24 | % | ALA4369978 | % | ||||
11. | ALA2012686 | 21 | Activity | 0 | ALA4369977 | Non-Toxic | ||||||
12. | ALA2012686 | 21 | Activity | 0 | ALA4369975 | Toxic | ||||||
13. | ALA2012686 | 21 | PPB | = | 94 | % | ALA4369974 | % | ||||
14. | ALA2012686 | 21 | PPB | = | 90 | % | ALA4369973 | % | ||||
15. | ALA2012686 | 21 | Ratio | = | 0.91 | ALA4369972 | ||||||
16. | ALA2012686 | 21 | Stability | = | 51 | % | ALA4369971 | % | ||||
17. | ALA2012686 | 21 | IC50 | > | 25 | uM | ALA4369970 | nM | Homo sapiens | |||
18. | ALA2012686 | 21 | IC50 | > | 25 | uM | ALA4369969 | nM | Homo sapiens | |||
19. | ALA2012686 | 21 | IC50 | > | 25 | uM | ALA4369968 | nM | Homo sapiens | |||
20. | ALA2012686 | 21 | F | = | 124 | % | ALA4369967 | % |