| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2022994 | rac-29 | GI50 | = | 200 | nM | ALA2330554 | nM | Homo sapiens | |||
| 2. | ALA2022994 | rac-29 | Ki(app) | = | 12.2 | nM | ALA2330556 | 7.91 | nM | Homo sapiens | ||
| 3. | ALA2022994 | rac-29 | Cmax | = | 1.2 | ug ml-1 | ALA2327403 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 4. | ALA2022994 | rac-29 | Tmax | = | 3.7 | hr | ALA2327404 | hr | Mus musculus | |||
| 5. | ALA2022994 | rac-29 | AUClast | = | 7.2 | microg.hr/mL | ALA2327402 | ng.hr.mL-1 | Mus musculus | |||
| 6. | ALA2022994 | rac-29 | C0 | = | 8.2 | ug ml-1 | ALA2327400 | ug ml-1 | Mus musculus | |||
| 7. | ALA2022994 | rac-29 | t1/2 | = | 6.5 | hr | ALA2327401 | hr | Mus musculus | |||
| 8. | ALA2022994 | rac-29 | Vd | = | 0.6 | L/Kg | ALA2327399 | L.kg-1 | Mus musculus | |||
| 9. | ALA2022994 | rac-29 | CL | = | 3.8 | ml/min.kg | ALA2327397 | mL.min-1.kg-1 | Mus musculus | |||
| 10. | ALA2022994 | rac-29 | AUClast | = | 13.1 | microg.hr/mL | ALA2327398 | ng.hr.mL-1 | Mus musculus | |||
| 11. | ALA2022994 | rac-29 | Activity | 0 | ALA2327396 | Active | ||||||
| 12. | ALA2022994 | rac-29 | Time | = | 28.7 | day | ALA2025103 | hr | ||||
| 13. | ALA2022994 | rac-29 | T/C | = | 26.3 | % | ALA2025102 | % | ||||
| 14. | ALA2022994 | rac-29 | GI50 | = | 144 | nM | ALA2024992 | nM | Homo sapiens | |||
| 15. | ALA2022994 | rac-29 | GI50 | = | 137 | nM | ALA2024991 | nM | Homo sapiens | |||
| 16. | ALA2022994 | rac-29 | GI50 | = | 38 | nM | ALA2024990 | nM | ||||
| 17. | ALA2022994 | rac-29 | GI50 | = | 99 | nM | ALA2024989 | nM | Homo sapiens | |||
| 18. | ALA2022994 | rac-29 | INH | 0 | ALA2024988 | Not Active | % | Homo sapiens | ||||
| 19. | ALA2022994 | rac-29 | INH | 0 | ALA2024987 | Not Active | % | Homo sapiens | ||||
| 20. | ALA2022994 | rac-29 | INH | 0 | ALA2024986 | Not Active | % | Homo sapiens |
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