# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2028983 | cyclo(Ppa-Tyr-Phe-Gln-Asn-Cys)-MeAla-Arg-Lys(N3PhCNH)-NH2 | logP | = | 1.62 | ALA876520 | ||||||
2. | ALA2028983 | cyclo(Ppa-Tyr-Phe-Gln-Asn-Cys)-MeAla-Arg-Lys(N3PhCNH)-NH2 | RA | = | 70 | % | ALA819411 | % | Rattus norvegicus | |||
3. | ALA2028983 | cyclo(Ppa-Tyr-Phe-Gln-Asn-Cys)-MeAla-Arg-Lys(N3PhCNH)-NH2 | pKd | = | 9.04 | ALA819412 | 9.04 | nM | Rattus norvegicus | |||
4. | ALA2028983 | cyclo(Ppa-Tyr-Phe-Gln-Asn-Cys)-MeAla-Arg-Lys(N3PhCNH)-NH2 | Kd | = | 0.92 | nM | ALA821119 | 9.04 | nM | Rattus norvegicus | ||
5. | ALA2028983 | cyclo(Ppa-Tyr-Phe-Gln-Asn-Cys)-MeAla-Arg-Lys(N3PhCNH)-NH2 | RA | = | 194 | % | ALA820961 | % | Rattus norvegicus | |||
6. | ALA2028983 | cyclo(Ppa-Tyr-Phe-Gln-Asn-Cys)-MeAla-Arg-Lys(N3PhCNH)-NH2 | pKd | = | 9.48 | ALA819412 | 9.48 | nM | Rattus norvegicus | |||
7. | ALA2028983 | cyclo(Ppa-Tyr-Phe-Gln-Asn-Cys)-MeAla-Arg-Lys(N3PhCNH)-NH2 | Kd | = | 0.33 | nM | ALA821119 | 9.48 | nM | Rattus norvegicus |