| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2030560 | 9 | IC50 | = | 0.23 | uM | ALA2061832 | 6.64 | nM | Toxoplasma gondii | ||
| 2. | ALA2030560 | 9 | Ki | = | 10 | uM | ALA2033711 | 5.00 | nM | Homo sapiens | ||
| 3. | ALA2030560 | 9 | Ki | > | 10 | uM | ALA2033710 | nM | Homo sapiens | |||
| 4. | ALA2030560 | 9 | Ki | = | 0.28 | uM | ALA2033709 | 6.55 | nM | |||
| 5. | ALA2030560 | 9 | Ki | = | 0.12 | uM | ALA2033708 | 6.92 | nM | |||
| 6. | ALA2030560 | 9 | Drug metabolism | 0 | ALA3532635 | metabolite_detected | Homo sapiens | |||||
| 7. | ALA2030560 | 9 | Drug metabolism | 0 | ALA3532633 | metabolite_detected | Homo sapiens | |||||
| 8. | ALA2030560 | 9 | CLint | < | 3 | microL/min/mg | ALA3301370 | mL.min-1.g-1 | ||||
| 9. | ALA2030560 | 9 | CLint | < | 3 | microL/min/1E6 cells | ALA3301371 | uL.min-1.(10^6cells)-1 | ||||
| 10. | ALA2030560 | 9 | PPB | 92.64 | % | ALA3301366 | % | |||||
| 11. | ALA2030560 | 9 | LogD7.4 | 2.29 | ALA3301363 | |||||||
| 12. | ALA2030560 | 9 | Activity | 0 | ALA4432267 | Active | Homo sapiens | |||||
| 13. | ALA2030560 | 9 | Kd | = | 13 | uM | ALA4432266 | 4.89 | nM | Homo sapiens | ||
| 14. | ALA2030560 | 9 | EC50 | > | 30 | uM | ALA2061821 | nM | ||||
| 15. | ALA2030560 | 9 | EC50 | > | 30 | uM | ALA2061822 | nM | Homo sapiens | |||
| 16. | ALA2030560 | 9 | Activity | 0 | ALA2061825 | Not Active | Cryptosporidium parvum | |||||
| 17. | ALA2030560 | 9 | Activity | 0 | ALA2061826 | Not Active | Toxoplasma gondii | |||||
| 18. | ALA2030560 | 9 | IC50 | = | 10 | uM | ALA2061829 | 5.00 | nM | Homo sapiens | ||
| 19. | ALA2030560 | 9 | IC50 | > | 10 | uM | ALA2061830 | nM | Homo sapiens | |||
| 20. | ALA2030560 | 9 | IC50 | = | 0.6 | uM | ALA2061831 | 6.22 | nM |
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