| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | F | = | 50 | % | ALA2033698 | % | Rattus norvegicus | |||
| 2. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Drug metabolism | 0 | ALA2033697 | Active | Rattus norvegicus | |||||
| 3. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Drug metabolism | 0 | ALA2033695 | Active | Mesocricetus auratus | |||||
| 4. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Drug metabolism | 0 | ALA2033693 | Active | Homo sapiens | |||||
| 5. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Drug metabolism | 0 | ALA2033692 | Not Active | Homo sapiens | |||||
| 6. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | F | = | 70 | % | ALA2033691 | % | Canis lupus familiaris | |||
| 7. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | beta t1/2 | = | 7 | hr | ALA2033690 | hr | Canis lupus familiaris | |||
| 8. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Vd | = | 1.66 | L/Kg | ALA2033689 | L.kg-1 | Canis lupus familiaris | |||
| 9. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | CL | = | 0.4 | L/hr/kg | ALA2033688 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 10. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Stability | = | 100 | % | ALA2033511 | % | ||||
| 11. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | IC50 | = | 0.31 | uM | ALA2033510 | 6.51 | nM | Hepacivirus hominis | ||
| 12. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | CC50 | = | 85 | uM | ALA2033509 | nM | Homo sapiens | |||
| 13. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | EC50 | = | 1.98 | uM | ALA2033508 | 5.70 | nM | Hepacivirus hominis | ||
| 14. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Drug metabolism | = | 29.7 | pmol | ALA3296476 | pmol | ||||
| 15. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Drug metabolism | = | 16.9 | pmol | ALA3297112 | pmol | Rattus norvegicus | |||
| 16. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Drug metabolism | = | 46.2 | pmol | ALA3297012 | pmol | Homo sapiens | |||
| 17. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Drug metabolism | = | 31.8 | pmol | ALA3296876 | pmol | ||||
| 18. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Activity | 0 | ALA3297011 | Toxic | Rattus norvegicus | |||||
| 19. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Activity | 0 | ALA3297007 | Non-toxic | Salmonella enterica subsp. enterica serovar Typhimurium | |||||
| 20. | ALA2031678 | 2, 2'-C-Me 4-aza-7,9-dideaza A | Activity | 0 | ALA3297006 | Non-toxic |
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