| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2036782 | 8c | IC50 | = | 22 | nM | ALA2039642 | 7.66 | nM | Homo sapiens | ||
| 2. | ALA2036782 | 8c | INH | 0 | ALA2039641 | Not Active | % | Homo sapiens | ||||
| 3. | ALA2036782 | 8c | INH | 0 | ALA2039640 | Not Active | % | Homo sapiens | ||||
| 4. | ALA2036782 | 8c | INH | 0 | ALA2039639 | Not Active | % | Homo sapiens | ||||
| 5. | ALA2036782 | 8c | INH | 0 | ALA2039638 | Not Active | % | Homo sapiens | ||||
| 6. | ALA2036782 | 8c | IC50 | = | 1.6 | uM | ALA2039637 | 5.80 | nM | |||
| 7. | ALA2036782 | 8c | IC50 | = | 0.2 | uM | ALA2039636 | 6.70 | nM | Rattus norvegicus | ||
| 8. | ALA2036782 | 8c | IC50 | = | 1.2 | uM | ALA2039635 | 5.92 | nM | Mus musculus | ||
| 9. | ALA2036782 | 8c | pA2 | = | 8.46 | ALA2039634 | 8.46 | nM | Homo sapiens | |||
| 10. | ALA2036782 | 8c | IC50 | = | 5.1 | nM | ALA2039633 | 8.29 | nM | Homo sapiens | ||
| 11. | ALA2036782 | 8c | Ratio IC50 | = | 10000 | ALA2039632 | ||||||
| 12. | ALA2036782 | 8c | IC50 | = | 60 | uM | ALA2039631 | 4.22 | nM | Homo sapiens | ||
| 13. | ALA2036782 | 8c | solubility | > | 3100 | uM | ALA2039630 | nM | ||||
| 14. | ALA2036782 | 8c | pKa | = | 7.8 | ALA2039629 | ||||||
| 15. | ALA2036782 | 8c | logP | = | 2.7 | ALA2039628 | ||||||
| 16. | ALA2036782 | 8c | logD | = | 2.21 | ALA2039627 | ||||||
| 17. | ALA2036782 | 8c | F | = | 83 | % | ALA2039626 | % | Canis lupus familiaris | |||
| 18. | ALA2036782 | 8c | F | = | 11 | % | ALA2039625 | % | Rattus norvegicus | |||
| 19. | ALA2036782 | 8c | t1/2 | = | 9.1 | hr | ALA2039624 | hr | Canis lupus familiaris | |||
| 20. | ALA2036782 | 8c | t1/2 | = | 3 | hr | ALA2039623 | hr | Rattus norvegicus |
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