| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2059300 | 25 | IC50 | = | 2.2 | nM | ALA2182642 | 8.66 | nM | Homo sapiens | ||
| 2. | ALA2059300 | 25 | IC50 | = | 19.9 | nM | ALA2182643 | 7.70 | nM | Homo sapiens | ||
| 3. | ALA2059300 | 25 | IC50 | = | 1.9 | uM | ALA2182644 | 5.72 | nM | Homo sapiens | ||
| 4. | ALA2059300 | 25 | IC50 | = | 0.19 | uM | ALA2182645 | 6.72 | nM | Homo sapiens | ||
| 5. | ALA2059300 | 25 | IC50 | = | 0.85 | uM | ALA2182646 | 6.07 | nM | Homo sapiens | ||
| 6. | ALA2059300 | 25 | IC50 | > | 25 | uM | ALA2182647 | nM | Homo sapiens | |||
| 7. | ALA2059300 | 25 | IC50 | = | 1 | uM | ALA2182648 | 6.00 | nM | Homo sapiens | ||
| 8. | ALA2059300 | 25 | FC | = | 15 | ALA2182649 | Mus musculus | |||||
| 9. | ALA2059300 | 25 | Activity | 0 | ALA2182650 | Dose-dependent effect | Mus musculus | |||||
| 10. | ALA2059300 | 25 | TGI | = | 91 | % | ALA2182651 | % | Homo sapiens | |||
| 11. | ALA2059300 | 25 | Kd | = | 1 | nM | ALA2182652 | 9.00 | nM | Homo sapiens | ||
| 12. | ALA2059300 | 25 | Activity | = | 27 | % | ALA2182653 | % | Homo sapiens | |||
| 13. | ALA2059300 | 25 | INH | = | 40 | % | ALA2182654 | % | Homo sapiens | |||
| 14. | ALA2059300 | 25 | Activity | = | 77 | % | ALA2182655 | % | Homo sapiens | |||
| 15. | ALA2059300 | 25 | CLH | = | 26 | uL/min | ALA2182664 | uL/min | ||||
| 16. | ALA2059300 | 25 | CL | = | 2.7 | L/hr/kg | ALA2182665 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 17. | ALA2059300 | 25 | Vdss | = | 1.5 | L/Kg | ALA2182666 | L.kg-1 | Rattus norvegicus | |||
| 18. | ALA2059300 | 25 | F | = | 77 | % | ALA2182667 | % | Rattus norvegicus | |||
| 19. | ALA2059300 | 25 | CL | = | 1.5 | L/hr/kg | ALA2182668 | mL.min-1.kg-1 | Mus musculus | |||
| 20. | ALA2059300 | 25 | Vdss | = | 1.3 | L/Kg | ALA2182669 | L.kg-1 | Mus musculus |
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