| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2069500 | 3 | Selectivity ratio | > | 1000 | ALA2072630 | ||||||
| 2. | ALA2069500 | 3 | Selectivity ratio | > | 1000 | ALA2072629 | ||||||
| 3. | ALA2069500 | 3 | Selectivity ratio | > | 1000 | ALA2072628 | ||||||
| 4. | ALA2069500 | 3 | Selectivity ratio | > | 1000 | ALA2072627 | ||||||
| 5. | ALA2069500 | 3 | Ki | = | 1.7 | nM | ALA2072626 | 8.77 | nM | Homo sapiens | ||
| 6. | ALA2069500 | 3 | F | = | 15 | % | ALA2072508 | % | Mus musculus | |||
| 7. | ALA2069500 | 3 | t1/2 | = | 0.14 | hr | ALA2072507 | hr | Mus musculus | |||
| 8. | ALA2069500 | 3 | CL | = | 95 | ml/min.kg | ALA2072506 | mL.min-1.kg-1 | Mus musculus | |||
| 9. | ALA2069500 | 3 | Vdss | = | 8.1 | L/Kg | ALA2072505 | L.kg-1 | Mus musculus | |||
| 10. | ALA2069500 | 3 | Cmax | = | 60 | nM | ALA2072504 | nM | Mus musculus | |||
| 11. | ALA2069500 | 3 | AUC/dose | = | 0.07 | uM.hr/mg | ALA2072503 | uM.hr/mg | Mus musculus | |||
| 12. | ALA2069500 | 3 | IC50 | = | 308 | nM | ALA2072502 | 6.51 | nM | Homo sapiens | ||
| 13. | ALA2069500 | 3 | IC50 | = | 77 | nM | ALA2072491 | 7.11 | nM | Homo sapiens | ||
| 14. | ALA2069500 | 3 | IC50 | = | 26 | nM | ALA2072490 | 7.58 | nM | Homo sapiens | ||
| 15. | ALA2069500 | 3 | IC50 | = | 0.8 | nM | ALA2072489 | 9.10 | nM | Homo sapiens | ||
| 16. | ALA2069500 | 3 | Ki | = | 0.08 | uM | ALA3583383 | 7.10 | nM | Homo sapiens | ||
| 17. | ALA2069500 | 3 | IC50 | = | 26.1 | nM | ALA3583382 | 7.58 | nM | Homo sapiens | ||
| 18. | ALA2069500 | 3 | IC50 | = | 0.8 | nM | ALA3583381 | 9.10 | nM | Homo sapiens |
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