| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2069501 | 4 | pKd | = | 8.69 | ALA2072631 | 8.69 | nM | Homo sapiens | |||
| 2. | ALA2069501 | 4 | Selectivity ratio | > | 400 | ALA2072630 | ||||||
| 3. | ALA2069501 | 4 | Selectivity ratio | > | 400 | ALA2072629 | ||||||
| 4. | ALA2069501 | 4 | Selectivity ratio | > | 400 | ALA2072628 | ||||||
| 5. | ALA2069501 | 4 | Selectivity ratio | > | 400 | ALA2072627 | ||||||
| 6. | ALA2069501 | 4 | F | = | 4 | % | ALA2072508 | % | Mus musculus | |||
| 7. | ALA2069501 | 4 | t1/2 | = | 0.54 | hr | ALA2072507 | hr | Mus musculus | |||
| 8. | ALA2069501 | 4 | CL | = | 31 | ml/min.kg | ALA2072506 | mL.min-1.kg-1 | Mus musculus | |||
| 9. | ALA2069501 | 4 | Vdss | = | 0.7 | L/Kg | ALA2072505 | L.kg-1 | Mus musculus | |||
| 10. | ALA2069501 | 4 | Cmax | = | 130 | nM | ALA2072504 | nM | Mus musculus | |||
| 11. | ALA2069501 | 4 | AUC/dose | = | 0.06 | uM.hr/mg | ALA2072503 | uM.hr/mg | Mus musculus | |||
| 12. | ALA2069501 | 4 | IC50 | = | 1526 | nM | ALA2072502 | 5.82 | nM | Homo sapiens | ||
| 13. | ALA2069501 | 4 | IC50 | = | 176 | nM | ALA2072491 | 6.75 | nM | Homo sapiens |
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