| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2074599 | E3040 glucuronide | Ki | = | 5.6 | uM | ALA2077552 | 5.25 | inhibitor [Ki=5.6uM] | nM | Homo sapiens | |
| 2. | ALA2074599 | E3040 glucuronide | Ki | = | 3.84 | uM | ALA2075074 | 5.42 | inhibitor [Ki=3.84uM] | nM | Rattus norvegicus | |
| 3. | ALA2074599 | E3040 glucuronide | Ki | = | 2.6 | uM | ALA2078011 | 5.58 | inhibitor [Ki=2.6uM] | nM | Rattus norvegicus | |
| 4. | ALA2074599 | E3040 glucuronide | Km | = | 5.7 | uM | ALA2075782 | substrate [Km=5.7uM] | nM | Rattus norvegicus | ||
| 5. | ALA2074599 | E3040 glucuronide | Activity | = | 76 | % | ALA2077939 | inhibitor [76% of control] | % | Homo sapiens | ||
| 6. | ALA2074599 | E3040 glucuronide | Activity | = | 11.1 | % | ALA2078015 | inhibitor [11.1 % of control] | % | Rattus norvegicus | ||
| 7. | ALA2074599 | E3040 glucuronide | Activity | 0 | ALA2076809 | substrate [] | Homo sapiens | |||||
| 8. | ALA2074599 | E3040 glucuronide | Activity | 0 | ALA2077551 | substrate [+] | Homo sapiens | |||||
| 9. | ALA2074599 | E3040 glucuronide | Activity | 0 | ALA2076292 | substrate [+] | Rattus norvegicus | |||||
| 10. | ALA2074599 | E3040 glucuronide | Activity | 0 | ALA2077358 | substrate [+] | Rattus norvegicus | |||||
| 11. | ALA2074599 | E3040 glucuronide | Km | = | 14.1 | uM | ALA2076879 | substrate [Km=14.1uM] | nM | Homo sapiens |
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