# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2086528 | 18d | IC50 | = | 10 | nM | ALA5225353 | 8.00 | nM | Homo sapiens | ||
2. | ALA2086528 | 18d | Ratio IC50 | = | 77 | ALA2091169 | Homo sapiens | |||||
3. | ALA2086528 | 18d | Ratio IC50 | = | 84 | ALA2091165 | ||||||
4. | ALA2086528 | 18d | Ratio IC50 | > | 8000 | ALA2091164 | ||||||
5. | ALA2086528 | 18d | Ratio IC50 | = | 340 | ALA2091163 | ||||||
6. | ALA2086528 | 18d | Ratio IC50 | = | 18 | ALA2091161 | ||||||
7. | ALA2086528 | 18d | Papp | = | 193 | nm/s | ALA2091173 | nm/s | Homo sapiens | |||
8. | ALA2086528 | 18d | Papp | = | 102 | nm/s | ALA2091172 | nm/s | Homo sapiens | |||
9. | ALA2086528 | 18d | CLH | = | 3203 | ml/min.kg | ALA2091214 | mL.min-1.kg-1 | Mus musculus | |||
10. | ALA2086528 | 18d | t1/2 | = | 248 | min | ALA2091213 | hr | Mus musculus | |||
11. | ALA2086528 | 18d | IC50 | = | 0.77 | uM | ALA2091168 | 6.11 | nM | Homo sapiens | ||
12. | ALA2086528 | 18d | IC50 | = | 0.016 | uM | ALA2091167 | 7.80 | nM | Mus musculus | ||
13. | ALA2086528 | 18d | IC50 | = | 0.84 | uM | ALA2091166 | 6.08 | nM | Homo sapiens | ||
14. | ALA2086528 | 18d | IC50 | = | 0.18 | uM | ALA2091160 | 6.75 | nM | Homo sapiens | ||
15. | ALA2086528 | 18d | IC50 | > | 80 | uM | ALA2091159 | nM | Homo sapiens | |||
16. | ALA2086528 | 18d | IC50 | = | 3.4 | uM | ALA2091158 | 5.47 | nM | Homo sapiens | ||
17. | ALA2086528 | 18d | IC50 | = | 0.01 | uM | ALA2091156 | 8.00 | nM | Homo sapiens | ||
18. | ALA2086528 | 18d | Fu | = | 2 | % | ALA2091171 | Homo sapiens | ||||
19. | ALA2086528 | 18d | Kinetic_solubility | = | 0.01 | mg/ml | ALA2091170 | ug.mL-1 |