# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2087456 | 21 | Activity | 0 | ALA2091654 | Not Active | Homo sapiens | |||||
2. | ALA2087456 | 21 | Activity | 0 | ALA2091653 | Not Active | Homo sapiens | |||||
3. | ALA2087456 | 21 | Activity | 0 | ALA2091652 | Not Active | Homo sapiens | |||||
4. | ALA2087456 | 21 | INH | = | -2 | % | ALA2091629 | % | Homo sapiens | |||
5. | ALA2087456 | 21 | INH | = | 21 | % | ALA2091628 | % | Homo sapiens | |||
6. | ALA2087456 | 21 | INH | = | 3 | % | ALA2091627 | % | Homo sapiens | |||
7. | ALA2087456 | 21 | Stability | = | 100 | % | ALA2091626 | % | Homo sapiens | |||
8. | ALA2087456 | 21 | permeability | > | 10 | ucm/s | ALA2091625 | ucm/s | ||||
9. | ALA2087456 | 21 | solubility | = | 133 | uM | ALA2091624 | nM | ||||
10. | ALA2087456 | 21 | IC50 | > | 30 | uM | ALA2091623 | nM | Homo sapiens | |||
11. | ALA2087456 | 21 | IC50 | > | 30 | uM | ALA2091475 | nM | Homo sapiens | |||
12. | ALA2087456 | 21 | IC50 | > | 30 | uM | ALA2091474 | nM | Homo sapiens | |||
13. | ALA2087456 | 21 | Emax | > | 90 | % | ALA2091473 | % | Rattus norvegicus | |||
14. | ALA2087456 | 21 | EC50 | = | 1.05 | uM | ALA2091472 | 5.98 | nM | Rattus norvegicus |