# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2088586 | 1 | INH | = | 0 | % | ALA2090356 | % | Rattus norvegicus | |||
2. | ALA2088586 | 1 | INH | = | 30 | % | ALA2090355 | % | Rattus norvegicus | |||
3. | ALA2088586 | 1 | F | = | 96 | % | ALA2090352 | % | Rattus norvegicus | |||
4. | ALA2088586 | 1 | AUC | = | 3.6 | uM.hr | ALA2090349 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
5. | ALA2088586 | 1 | CL | = | 11.6 | ml/min.kg | ALA2090346 | mL.min-1.kg-1 | Rattus norvegicus | |||
6. | ALA2088586 | 1 | t1/2 | = | 1.1 | hr | ALA2090343 | hr | Rattus norvegicus | |||
7. | ALA2088586 | 1 | EC50 | > | 30000 | nM | ALA2090341 | nM | Homo sapiens | |||
8. | ALA2088586 | 1 | IC50 | = | 26 | nM | ALA2090340 | 7.58 | nM | Homo sapiens | ||
9. | ALA2088586 | 1 | IC50 | = | 29 | nM | ALA2090339 | 7.54 | nM | Homo sapiens | ||
10. | ALA2088586 | 1 | Ratio IC50 | = | 18 | ALA2090338 | ||||||
11. | ALA2088586 | 1 | IC50 | = | 86 | nM | ALA2090337 | 7.07 | nM | Mus musculus | ||
12. | ALA2088586 | 1 | IC50 | = | 4.7 | nM | ALA2090336 | 8.33 | nM | Mus musculus |