# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2130955 | SID85201013 | Drug recovery | > | 95 | % | ALA5115447 | % | ||||
2. | ALA2130955 | SID85201013 | Drug recovery | = | 87 | % | ALA5115446 | % | ||||
3. | ALA2130955 | SID85201013 | Drug recovery | = | 89 | % | ALA5115445 | % | ||||
4. | ALA2130955 | SID85201013 | solubility | = | 3.4 | uM | ALA5115444 | nM | ||||
5. | ALA2130955 | SID85201013 | Papp | = | 4.1 | 10^-6 cm/s | ALA5115443 | 10^-6 cm/s | ||||
6. | ALA2130955 | SID85201013 | Papp | = | 4.6 | 10^-6 cm/s | ALA5115442 | 10^-6 cm/s | ||||
7. | ALA2130955 | SID85201013 | PPB | > | 95 | % | ALA5115441 | % | ||||
8. | ALA2130955 | SID85201013 | logP | = | 4.06 | ALA5115440 | ||||||
9. | ALA2130955 | SID85201013 | IC50 | = | 1.1 | uM | ALA5115439 | 5.96 | nM | Homo sapiens | ||
10. | ALA2130955 | SID85201013 | IC50 | = | 1.9 | uM | ALA5115438 | 5.72 | nM | Homo sapiens | ||
11. | ALA2130955 | SID85201013 | INH | < | 25 | % | ALA5115437 | % | Homo sapiens | |||
12. | ALA2130955 | SID85201013 | IC50 | = | 50 | uM | ALA5115436 | 4.30 | nM | Homo sapiens | ||
13. | ALA2130955 | SID85201013 | INH | < | 25 | % | ALA5115435 | % | Homo sapiens | |||
14. | ALA2130955 | SID85201013 | IC50 | = | 50 | uM | ALA5115434 | 4.30 | nM | Homo sapiens | ||
15. | ALA2130955 | SID85201013 | IC50 | = | 0.87 | uM | ALA5115433 | 6.06 | nM | Homo sapiens | ||
16. | ALA2130955 | SID85201013 | IC50 | = | 0.76 | uM | ALA5115432 | 6.12 | nM | Homo sapiens | ||
17. | ALA2130955 | SID85201013 | IC50 | = | 7.6 | uM | ALA5115431 | 5.12 | nM | |||
18. | ALA2130955 | SID85201013 | IC50 | = | 0.71 | uM | ALA5115430 | 6.15 | nM | |||
19. | ALA2130955 | SID85201013 | IC50 | = | 4.3 | uM | ALA5115429 | 5.37 | nM | |||
20. | ALA2130955 | SID85201013 | IC50 | = | 1.4 | uM | ALA5115428 | 5.85 | nM |