# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2135857 | SID17389435 | Stability | 0 | ALA3283238 | Stable | % | |||||
2. | ALA2135857 | SID17389435 | Stability | 0 | ALA3283237 | Stable | % | |||||
3. | ALA2135857 | SID17389435 | Stability | 0 | ALA3283239 | Stable | % | |||||
4. | ALA2135857 | SID17389435 | t1/2 | = | 24 | hr | ALA3283526 | hr | ||||
5. | ALA2135857 | SID17389435 | pKa | = | 8.6 | ALA3283525 | ||||||
6. | ALA2135857 | SID17389435 | INH | 0 | ALA3283524 | Active | % | |||||
7. | ALA2135857 | SID17389435 | ED50 | = | 1.21 | 10'-4M | ALA3283523 | 10'-4M | ||||
8. | ALA2135857 | SID17389435 | ED50 | = | 5.05 | 10'-4M | ALA3283249 | 10'-4M | ||||
9. | ALA2135857 | SID17389435 | Drug degradation | = | 0.06 | 10'-8mol/min | ALA3283248 | 10'-8mol/min | Homo sapiens | |||
10. | ALA2135857 | SID17389435 | Drug degradation | = | 0.07 | 10'-8mol/min | ALA3283247 | 10'-8mol/min | Homo sapiens | |||
11. | ALA2135857 | SID17389435 | Drug degradation | = | 1.75 | 10'-8mol/min | ALA3283246 | 10'-8mol/min | ||||
12. | ALA2135857 | SID17389435 | INH | 0 | ALA3283245 | Active | % | Rattus norvegicus | ||||
13. | ALA2135857 | SID17389435 | INH | 0 | ALA3283244 | Active | % | Rattus norvegicus | ||||
14. | ALA2135857 | SID17389435 | INH | 0 | ALA3283243 | Active | % | Rattus norvegicus | ||||
15. | ALA2135857 | SID17389435 | INH | 0 | ALA3283240 | Active | % | Rattus norvegicus | ||||
16. | ALA2135857 | SID17389435 | I50 | = | 5.02 | 10'-4M | ALA3283242 | nM | Rattus norvegicus | |||
17. | ALA2135857 | SID17389435 | INH | 0 | ALA3283234 | Not Active | % | Rattus norvegicus | ||||
18. | ALA2135857 | SID17389435 | Stability | 0 | ALA3283236 | Stable | % | |||||
19. | ALA2135857 | SID17389435 | Stability | 0 | ALA3283235 | Unstable | % | |||||
20. | ALA2135857 | SID17389435 | Potency | 74.978 | uM | ALA2114835 | inconclusive | nM | Homo sapiens |