| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2146755 | 5 | IC50 | = | 66 | nM | ALA3705830 | 7.18 | 311055 | nM | Homo sapiens | |
| 2. | ALA2146755 | 5 | IC50 | = | 0.052 | uM | ALA4427467 | 7.28 | nM | Homo sapiens | ||
| 3. | ALA2146755 | 5 | IC50 | = | 0.007 | uM | ALA4427468 | 8.15 | nM | Homo sapiens | ||
| 4. | ALA2146755 | 5 | Ratio IC50 | = | 0.13 | ALA4427469 | ||||||
| 5. | ALA2146755 | 5 | F | = | 14 | % | ALA2148636 | % | Rattus norvegicus | |||
| 6. | ALA2146755 | 5 | AUC/dose | = | 0.023 | uM.hr.kg/mg | ALA2148635 | uM.hr.kg/mg | Rattus norvegicus | |||
| 7. | ALA2146755 | 5 | t1/2 | = | 1.9 | hr | ALA2148634 | hr | Rattus norvegicus | |||
| 8. | ALA2146755 | 5 | CL | = | 261 | L/Kg | ALA2148633 | L/Kg | Rattus norvegicus | |||
| 9. | ALA2146755 | 5 | INH | < | 50 | % | ALA2148632 | % | Homo sapiens | |||
| 10. | ALA2146755 | 5 | INH | < | 50 | % | ALA2148631 | % | Homo sapiens | |||
| 11. | ALA2146755 | 5 | IC50 | = | 0.024 | uM | ALA2148630 | 7.62 | nM | Homo sapiens | ||
| 12. | ALA2146755 | 5 | IC50 | > | 100 | uM | ALA2148628 | nM | Homo sapiens | |||
| 13. | ALA2146755 | 5 | IC50 | > | 100 | uM | ALA2148627 | nM | Homo sapiens | |||
| 14. | ALA2146755 | 5 | Ratio IC50 | = | 10 | ALA2148629 | ||||||
| 15. | ALA2146755 | 5 | IC50 | = | 0.005 | uM | ALA2148626 | 8.30 | nM | Homo sapiens | ||
| 16. | ALA2146755 | 5 | IC50 | = | 0.052 | uM | ALA2148625 | 7.28 | nM | Homo sapiens |
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