| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2147472 | 19a | INH | = | 68 | % | ALA3858677 | % | ||||
| 2. | ALA2147472 | 19a | Activity | 0 | ALA3858591 | Non-Toxic | Rattus norvegicus | |||||
| 3. | ALA2147472 | 19a | Activity | = | 4.2 | % | ALA3858604 | % | ||||
| 4. | ALA2147472 | 19a | Activity | = | 4.1 | % | ALA3858605 | % | ||||
| 5. | ALA2147472 | 19a | Fu | = | 0.2 | % | ALA3858586 | |||||
| 6. | ALA2147472 | 19a | logP | = | 4.8 | ALA3858585 | ||||||
| 7. | ALA2147472 | 19a | solubility | < | 1 | ug ml-1 | ALA3858584 | ug.mL-1 | ||||
| 8. | ALA2147472 | 19a | Stability | = | 100 | % | ALA3858583 | % | ||||
| 9. | ALA2147472 | 19a | Stability | = | 95 | % | ALA3858582 | % | ||||
| 10. | ALA2147472 | 19a | Stability | = | 90 | % | ALA3858581 | % | ||||
| 11. | ALA2147472 | 19a | Ki | = | 16.9 | nM | ALA3858580 | 7.77 | nM | |||
| 12. | ALA2147472 | 19a | Activity | = | 14.7 | % | ALA3858614 | % | ||||
| 13. | ALA2147472 | 19a | Activity | = | 14.3 | % | ALA3858613 | % | ||||
| 14. | ALA2147472 | 19a | INH | 0 | ALA3858596 | % | Homo sapiens | |||||
| 15. | ALA2147472 | 19a | AUC | = | 11.5 | uM.hr | ALA3858652 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 16. | ALA2147472 | 19a | AUC | = | 5.2 | uM.hr | ALA3858654 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 17. | ALA2147472 | 19a | AUC | = | 22.1 | uM.hr | ALA3858656 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 18. | ALA2147472 | 19a | t1/2 | > | 24 | hr | ALA3858658 | hr | ||||
| 19. | ALA2147472 | 19a | t1/2 | = | 16 | hr | ALA3858659 | hr | ||||
| 20. | ALA2147472 | 19a | t1/2 | = | 37 | hr | ALA3858660 | hr |
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