| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2152768 | 3 | Ratio IC50 | = | 340 | ALA3395887 | ||||||
| 2. | ALA2152768 | 3 | IC50 | = | 3.8 | nM | ALA3395878 | 8.42 | nM | Homo sapiens | ||
| 3. | ALA2152768 | 3 | IC50 | = | 0.003 | uM | ALA2217262 | 8.46 | nM | Homo sapiens | ||
| 4. | ALA2152768 | 3 | Ratio IC50 | > | 350 | ALA2217276 | ||||||
| 5. | ALA2152768 | 3 | IC50 | = | 0.041 | uM | ALA2217317 | 7.39 | nM | Homo sapiens | ||
| 6. | ALA2152768 | 3 | INH | = | -6.9 | % | ALA2157247 | % | Homo sapiens | |||
| 7. | ALA2152768 | 3 | INH | = | 6.4 | % | ALA2157246 | % | Homo sapiens | |||
| 8. | ALA2152768 | 3 | INH | = | 8.7 | % | ALA2157245 | % | Homo sapiens | |||
| 9. | ALA2152768 | 3 | INH | = | 8.6 | % | ALA2157244 | % | Homo sapiens | |||
| 10. | ALA2152768 | 3 | INH | 0 | ALA2155530 | tde | % | Homo sapiens | ||||
| 11. | ALA2152768 | 3 | F | = | 90 | % | ALA2155529 | % | Rattus norvegicus | |||
| 12. | ALA2152768 | 3 | F | = | 80 | % | ALA2155528 | % | Mus musculus | |||
| 13. | ALA2152768 | 3 | PPB | = | 86 | % | ALA2155527 | % | Homo sapiens | |||
| 14. | ALA2152768 | 3 | t1/2 | = | 4.8 | hr | ALA2157757 | hr | Rattus norvegicus | |||
| 15. | ALA2152768 | 3 | t1/2 | = | 5 | hr | ALA2157756 | hr | Mus musculus | |||
| 16. | ALA2152768 | 3 | AUC | = | 46 | uM.hr | ALA2157755 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 17. | ALA2152768 | 3 | AUC | = | 63 | uM.hr | ALA2157754 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 18. | ALA2152768 | 3 | Cmax | = | 4.7 | uM | ALA2157753 | nM | Rattus norvegicus | |||
| 19. | ALA2152768 | 3 | Cmax | = | 14 | uM | ALA2157752 | nM | Mus musculus | |||
| 20. | ALA2152768 | 3 | t1/2 | = | 3.8 | hr | ALA2157751 | hr | Rattus norvegicus |
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