# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2153440 | 2d | IC50 | = | 40 | nM | ALA2156127 | 7.40 | nM | Homo sapiens | ||
2. | ALA2153440 | 2d | IC50 | = | 115 | nM | ALA2155423 | 6.94 | nM | Rattus norvegicus | ||
3. | ALA2153440 | 2d | Cp | = | 15 | uM | ALA2155434 | uM | Rattus norvegicus | |||
4. | ALA2153440 | 2d | AUC | = | 119 | uM.hr | ALA2155431 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
5. | ALA2153440 | 2d | Tmax | = | 3.3 | hr | ALA2155430 | hr | Rattus norvegicus | |||
6. | ALA2153440 | 2d | Cmax | = | 17.8 | uM | ALA2155429 | nM | Rattus norvegicus | |||
7. | ALA2153440 | 2d | beta t1/2 | = | 1.2 | hr | ALA2155428 | hr | Rattus norvegicus | |||
8. | ALA2153440 | 2d | Vdss | = | 0.2 | L/Kg | ALA2155427 | L.kg-1 | Rattus norvegicus | |||
9. | ALA2153440 | 2d | CL | = | 4.4 | ml/min.kg | ALA2155426 | mL.min-1.kg-1 | Rattus norvegicus | |||
10. | ALA2153440 | 2d | Cmax | = | 82.7 | uM | ALA2155425 | nM | Rattus norvegicus | |||
11. | ALA2153440 | 2d | IC50 | = | 7 | uM | ALA2155424 | 5.16 | nM | Homo sapiens | ||
12. | ALA2153440 | 2d | CLH | = | 0.22 | nmol/min/mg | ALA2155421 | nmol/min/mg | Rattus norvegicus |